Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50001696
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50000788([17-(2,3-3H-2-propenyl)]-4, 5a -epoxy-3,14-dihydro...)
Affinity DataKi:  1.10nMAssay Description:The ability to displace [3H]-naloxone from the Opioid receptor mu isolated from rat brain membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017412(CHEMBL345120 | Furan-2-carboxylic acid (1-phenethy...)
Affinity DataKi:  1.90nMAssay Description:The ability to displace [3H]-naloxone from the Opioid receptor mu isolated from rat brain membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50008984(N-(1-Phenethyl-piperidin-4-yl)-N-phenyl-propionami...)
Affinity DataKi:  2.20nMAssay Description:The ability to displace [3H]-naloxone from the Opioid receptor mu isolated from rat brain membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017406(CHEMBL162700 | Furan-3-carboxylic acid benzo[1,2,5...)
Affinity DataKi:  2.60nMAssay Description:The ability to displace [3H]-naloxone from the Opioid receptor mu isolated from rat brain membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017416(CHEMBL347188 | Furan-2-carboxylic acid (4-methyl-p...)
Affinity DataKi:  4.10nMAssay Description:The ability to displace [3H]-naloxone from the Opioid receptor mu isolated from rat brain membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017404(Mirfentanil hydrochloride | CHEMBL161084 | Furan-2...)
Affinity DataKi:  7.5nMAssay Description:The ability to displace [3H]-naloxone from the Opioid receptor mu isolated from rat brain membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017420(CHEMBL157922 | Furan-2-carboxylic acid (1-phenethy...)
Affinity DataKi:  7.70nMAssay Description:The ability to displace [3H]-naloxone from the Opioid receptor mu isolated from rat brain membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017403(CHEMBL161442 | Furan-2-carboxylic acid (1-phenethy...)
Affinity DataKi:  8.40nMAssay Description:The ability to displace [3H]naloxone from the opioid receptor mu isolated from rat brain membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017405(CHEMBL161511 | 2-Methoxy-N-(1-phenethyl-piperidin-...)
Affinity DataKi:  13nMAssay Description:The ability to displace [3H]-naloxone from the Opioid receptor mu isolated from rat brain membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017411(CHEMBL158857 | Furan-2-carboxylic acid (1-phenethy...)
Affinity DataKi:  14nMAssay Description:The ability to displace [3H]-naloxone from the Opioid receptor mu isolated from rat brain membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017410(CHEMBL161021 | 2-Methoxy-N-(1-phenethyl-piperidin-...)
Affinity DataKi:  16nMAssay Description:The ability to displace [3H]-naloxone from the Opioid receptor mu isolated from rat brain membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017409(CHEMBL161023 | Furan-2-carboxylic acid (6-chloro-p...)
Affinity DataKi:  19nMAssay Description:The ability to displace [3H]-naloxone from the Opioid receptor mu isolated from rat brain membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017414(CHEMBL161147 | Furan-3-carboxylic acid (2-chloro-p...)
Affinity DataKi:  21nMAssay Description:The ability to displace [3H]-naloxone from the Opioid receptor mu isolated from rat brain membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017413(CHEMBL161082 | Furan-2-carboxylic acid (2-chloro-p...)
Affinity DataKi:  22nMAssay Description:The ability to displace [3H]-naloxone from the Opioid receptor mu isolated from rat brain membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017402(CHEMBL158856 | Furan-3-carboxylic acid (1-phenethy...)
Affinity DataKi:  35nMAssay Description:The ability to displace [3H]-naloxone from the Opioid receptor mu isolated from rat brain membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017408(CHEMBL351672 | Furan-3-carboxylic acid (1-phenethy...)
Affinity DataKi: >100nMAssay Description:The ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from rat brain membrane; >= no displacementMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017397(CHEMBL423430 | 1-Phenethyl-piperidin-4-ylamine)
Affinity DataKi: >100nMAssay Description:The ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from rat brain membrane; >= no displacementMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017407(CHEMBL161057 | Furan-3-carboxylic acid (6-chloro-p...)
Affinity DataKi: >100nMAssay Description:The ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from rat brain membrane; >= absolutely no % changeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017401(CHEMBL422180 | Furan-3-carboxylic acid (1-phenethy...)
Affinity DataKi: >100nMAssay Description:The ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from rat brain membrane; >= no displacementMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017400(CHEMBL352442 | Furan-3-carboxylic acid (2-chloro-p...)
Affinity DataKi: >100nMAssay Description:The ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from rat brain membrane; >= no displacementMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017415(CHEMBL161487 | Furan-2-carboxylic acid morpholin-4...)
Affinity DataKi: >100nMAssay Description:The ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from rat brain membrane; >= no displacementMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017418(CHEMBL161512 | Furan-2-carboxylic acid (1-phenethy...)
Affinity DataKi: >100nMAssay Description:The ability to displace [3H]naloxone from the opioid receptor mu isolated from rat brain membrane; >= no displacementMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017417(CHEMBL347810 | Furan-3-carboxylic acid (6-chloro-p...)
Affinity DataKi: >100nMAssay Description:The ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from rat brain membrane; >= no displacementMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017419(CHEMBL161217 | 2-Methoxy-N-(1-phenethyl-piperidin-...)
Affinity DataKi: >100nMAssay Description:The ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from rat brain membrane; >= no displacementMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017398(CHEMBL159123 | 2-Methoxy-N-morpholin-4-yl-N-(1-phe...)
Affinity DataKi: >100nMAssay Description:The ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from rat brain membrane; >= no displacementMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Boc Technical Center

Curated by ChEMBL
LigandPNGBDBM50017399(CHEMBL161280 | N-(6-Chloro-pyrimidin-4-yl)-2-metho...)
Affinity DataKi:  214nMAssay Description:The ability to displace [3H]-naloxone from the Opioid receptor mu isolated from rat brain membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed