Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50046276
TargetBromodomain-containing protein 4(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 8nMAssay Description:Inhibition of BRD4 bromodomain-1 (unknown origin) by europium based LANCE TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50380682(CHEMBL2017291 | I-BET151 (16))
Affinity DataIC50: 107nMAssay Description:Inhibition of BRD4 bromodomain-1 (unknown origin) by europium based LANCE TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50103502(CHEMBL3398341)
Affinity DataIC50: 427nMAssay Description:Inhibition of BRD4 bromodomain-1 (unknown origin) by europium based LANCE TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208 | US2...)
Affinity DataIC50: 645nMAssay Description:Inhibition of BRD4 bromodomain-1 (unknown origin) by europium based LANCE TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50103495(CHEMBL3398340)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of BRD4 bromodomain-1 (unknown origin) by europium based LANCE TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50103496(CHEMBL3398328)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of BRD4 bromodomain-1 (unknown origin) by europium based LANCE TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50103497(CHEMBL3398326)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of BRD4 bromodomain-1 (unknown origin) by europium based LANCE TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50103498(CHEMBL3398339)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of BRD4 bromodomain-1 (unknown origin) by europium based LANCE TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50103500(CHEMBL3398325)
Affinity DataIC50: 1.79E+4nMAssay Description:Inhibition of BRD4 bromodomain-1 (unknown origin) by europium based LANCE TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50103491(CHEMBL3398338)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of BRD4 bromodomain-1 (unknown origin) by europium based LANCE TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50103499(CHEMBL3398337)
Affinity DataIC50: 2.97E+4nMAssay Description:Inhibition of BRD4 bromodomain-1 (unknown origin) by europium based LANCE TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM85771(6-(N-benzoylamino)purine, 2)
Affinity DataIC50: 3.42E+4nMAssay Description:Inhibition of BRD4 bromodomain-1 (unknown origin) by europium based LANCE TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50103493(CHEMBL3398332)
Affinity DataIC50: 3.45E+4nMAssay Description:Inhibition of BRD4 bromodomain-1 (unknown origin) by europium based LANCE TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50103492(CHEMBL3398334)
Affinity DataIC50: 6.30E+4nMAssay Description:Inhibition of BRD4 bromodomain-1 (unknown origin) by europium based LANCE TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50103494(CHEMBL3398330)
Affinity DataIC50: 7.86E+4nMAssay Description:Inhibition of BRD4 bromodomain-1 (unknown origin) by europium based LANCE TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed