Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50048823
LigandPNGBDBM50228318(CHEMBL279807)
Affinity DataKi:  0.355nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in rat cerebral cortical membrane, determined using [3H]- yohimbine as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2019
Entry Details Article
PubMed
LigandPNGBDBM50228316(CHEMBL62912)
Affinity DataKi:  0.661nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in rat cerebral cortical membrane, determined using [3H]- yohimbine as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2019
Entry Details Article
PubMed
LigandPNGBDBM50019848(CHEMBL10316 | Idazoxan | US8633208, Idazoxan | 4,5...)
Affinity DataKi:  11nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in rat cerebral cortical membrane, determined using [3H]- yohimbine as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2019
Entry Details Article
PubMed
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  13nMAssay Description:Binding affinity against Alpha-2 adrenergic receptor in rat cerebral cortical membrane, determined using [3H]- yohimbine as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2019
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  398nMAssay Description:Binding affinity against Alpha-1 adrenergic receptor in rat cerebral cortical membrane, determined using [3H]-prazosin as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2019
Entry Details Article
PubMed
LigandPNGBDBM50228317(CHEMBL62833)
Affinity DataKi:  479nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in rat cerebral cortical membrane, determined using [3H]- yohimbine as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2019
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50019848(CHEMBL10316 | Idazoxan | US8633208, Idazoxan | 4,5...)
Affinity DataKi:  794nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in rat cerebral cortical membrane, determined using [3H]prazosin as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2019
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50228318(CHEMBL279807)
Affinity DataKi:  5.13E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in rat cerebral cortical membrane, determined using [3H]prazosin as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2019
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50228317(CHEMBL62833)
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in rat cerebral cortical membrane, determined using [3H]prazosin as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2019
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50228316(CHEMBL62912)
Affinity DataKi:  1.02E+4nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in rat cerebral cortical membrane, determined using [3H]prazosin as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2019
Entry Details Article
PubMed