Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50045497
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065241(CHEMBL2207044)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 5 mins before substrate addition by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065108(CHEMBL3403818)
Affinity DataIC50: 1.60E+3nMAssay Description:Time-dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate compound preincubated for 30 mins with NADPH before substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065197(CHEMBL3403824)
Affinity DataIC50: 1.90E+3nMAssay Description:Time-dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate compound preincubated for 30 mins with NADPH before substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065109(CHEMBL3403819)
Affinity DataIC50: 2.70E+3nMAssay Description:Time-dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate compound preincubated for 30 mins with NADPH before substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065193(CHEMBL3403820)
Affinity DataIC50: 2.70E+3nMAssay Description:Time-dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate compound preincubated for 30 mins with NADPH before substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065193(CHEMBL3403820)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 5 mins before substrate addition by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065194(CHEMBL3403821)
Affinity DataIC50: 3.20E+3nMAssay Description:Time-dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate compound preincubated for 30 mins with NADPH before substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065203(CHEMBL2206994)
Affinity DataIC50: 3.90E+3nMAssay Description:Time-dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate compound preincubated for 30 mins with NADPH before substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065194(CHEMBL3403821)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 5 mins before substrate addition by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065109(CHEMBL3403819)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 5 mins before substrate addition by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065197(CHEMBL3403824)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 5 mins before substrate addition by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065196(CHEMBL3403823)
Affinity DataIC50: 7.70E+3nMAssay Description:Time-dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate compound preincubated for 30 mins with NADPH before substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065198(CHEMBL3403825)
Affinity DataIC50: 7.80E+3nMAssay Description:Time-dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate compound preincubated for 30 mins with NADPH before substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065199(CHEMBL3403826)
Affinity DataIC50: 1.10E+4nMAssay Description:Time-dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate compound preincubated for 30 mins with NADPH before substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065203(CHEMBL2206994)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 5 mins before substrate addition by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065108(CHEMBL3403818)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 5 mins before substrate addition by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065196(CHEMBL3403823)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 5 mins before substrate addition by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065199(CHEMBL3403826)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 5 mins before substrate addition by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065195(CHEMBL3403822)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 5 mins before substrate addition by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065195(CHEMBL3403822)
Affinity DataIC50: 1.60E+4nMAssay Description:Time-dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate compound preincubated for 30 mins with NADPH before substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065200(CHEMBL3403827)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 5 mins before substrate addition by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065200(CHEMBL3403827)
Affinity DataIC50: 1.70E+4nMAssay Description:Time-dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate compound preincubated for 30 mins with NADPH before substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065198(CHEMBL3403825)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 5 mins before substrate addition by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065201(CHEMBL3403816)
Affinity DataIC50: 2.50E+4nMAssay Description:Time-dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate compound preincubated for 30 mins with NADPH before substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065202(CHEMBL3403815)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 5 mins before substrate addition by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065202(CHEMBL3403815)
Affinity DataIC50: 2.50E+4nMAssay Description:Time-dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate compound preincubated for 30 mins with NADPH before substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065201(CHEMBL3403816)
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 5 mins before substrate addition by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065236(CHEMBL3403817)
Affinity DataIC50: 5.40E+4nMAssay Description:Time-dependent inhibition of CYP3A4 in human liver microsomes using midazolam as substrate compound preincubated for 30 mins with NADPH before substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Satori Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50065236(CHEMBL3403817)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 5 mins before substrate addition by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed