Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50045862
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086602(CHEMBL3426300)
Affinity DataEC50:  0.0450nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP accumulation incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086603(CHEMBL3426241)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP accumulation incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50301953((3S,6S,9S,12S,15S,21S)-21-(2-((S)-2-amino-3-(1H-im...)
Affinity DataEC50:  0.190nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP accumulation incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086603(CHEMBL3426241)
Affinity DataKi:  0.570nMAssay Description:Displacement of [125I]-17 from human GLP-1R expressed in CHO cell membranes incubated for 120 mins by scintillation counting based radioligand bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50301953((3S,6S,9S,12S,15S,21S)-21-(2-((S)-2-amino-3-(1H-im...)
Affinity DataKi:  0.660nMAssay Description:Displacement of [125I]-17 from human GLP-1R expressed in CHO cell membranes incubated for 120 mins by scintillation counting based radioligand bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086599(CHEMBL3426297)
Affinity DataEC50:  0.730nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP accumulation incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086598(CHEMBL3426296)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP accumulation incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086602(CHEMBL3426300)
Affinity DataKi:  6nMAssay Description:Displacement of [125I]-17 from human GLP-1R expressed in CHO cell membranes incubated for 120 mins by scintillation counting based radioligand bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086588(CHEMBL3426243)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP accumulation incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086588(CHEMBL3426243)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]-17 from human GLP-1R expressed in CHO cell membranes incubated for 120 mins by scintillation counting based radioligand bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086599(CHEMBL3426297)
Affinity DataKi:  41nMAssay Description:Displacement of [125I]-17 from human GLP-1R expressed in CHO cell membranes incubated for 120 mins by scintillation counting based radioligand bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086587(CHEMBL3426242)
Affinity DataKi:  59nMAssay Description:Displacement of [125I]-17 from human GLP-1R expressed in CHO cell membranes incubated for 120 mins by scintillation counting based radioligand bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086587(CHEMBL3426242)
Affinity DataEC50:  68nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP accumulation incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086595(CHEMBL3426293)
Affinity DataEC50:  81nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP accumulation incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086589(CHEMBL3426244)
Affinity DataEC50:  95nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP accumulation incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086597(CHEMBL3426295)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP accumulation incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086598(CHEMBL3426296)
Affinity DataKi:  130nMAssay Description:Displacement of [125I]-17 from human GLP-1R expressed in CHO cell membranes incubated for 120 mins by scintillation counting based radioligand bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086594(CHEMBL3426292)
Affinity DataEC50:  190nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP accumulation incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086601(CHEMBL3426299)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP accumulation incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086589(CHEMBL3426244)
Affinity DataKi:  300nMAssay Description:Displacement of [125I]-17 from human GLP-1R expressed in CHO cell membranes incubated for 120 mins by scintillation counting based radioligand bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086590(CHEMBL3426245)
Affinity DataEC50:  320nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP accumulation incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086591(CHEMBL3426246)
Affinity DataKi:  320nMAssay Description:Displacement of [125I]-17 from human GLP-1R expressed in CHO cell membranes incubated for 120 mins by scintillation counting based radioligand bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086600(CHEMBL3426298)
Affinity DataEC50:  390nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP accumulation incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086591(CHEMBL3426246)
Affinity DataEC50:  430nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP accumulation incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086595(CHEMBL3426293)
Affinity DataKi:  550nMAssay Description:Displacement of [125I]-17 from human GLP-1R expressed in CHO cell membranes incubated for 120 mins by scintillation counting based radioligand bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086593(CHEMBL3426291)
Affinity DataEC50:  600nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP accumulation incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086592(CHEMBL3426247)
Affinity DataEC50:  670nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP accumulation incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086596(CHEMBL3426294)
Affinity DataEC50:  730nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP accumulation incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086594(CHEMBL3426292)
Affinity DataKi:  980nMAssay Description:Displacement of [125I]-17 from human GLP-1R expressed in CHO cell membranes incubated for 120 mins by scintillation counting based radioligand bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086590(CHEMBL3426245)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [125I]-17 from human GLP-1R expressed in CHO cell membranes incubated for 120 mins by scintillation counting based radioligand bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086601(CHEMBL3426299)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [125I]-17 from human GLP-1R expressed in CHO cell membranes incubated for 120 mins by scintillation counting based radioligand bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086593(CHEMBL3426291)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [125I]-17 from human GLP-1R expressed in CHO cell membranes incubated for 120 mins by scintillation counting based radioligand bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086600(CHEMBL3426298)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [125I]-17 from human GLP-1R expressed in CHO cell membranes incubated for 120 mins by scintillation counting based radioligand bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086592(CHEMBL3426247)
Affinity DataKi: >3.10E+3nMAssay Description:Displacement of [125I]-17 from human GLP-1R expressed in CHO cell membranes incubated for 120 mins by scintillation counting based radioligand bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086597(CHEMBL3426295)
Affinity DataKi:  4.80E+3nMAssay Description:Displacement of [125I]-17 from human GLP-1R expressed in CHO cell membranes incubated for 120 mins by scintillation counting based radioligand bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50086596(CHEMBL3426294)
Affinity DataKi: >8.00E+3nMAssay Description:Displacement of [125I]-17 from human GLP-1R expressed in CHO cell membranes incubated for 120 mins by scintillation counting based radioligand bindin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed