Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50045968
TargetMethylosome protein 50/Protein arginine N-methyltransferase 5(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50089221(CHEMBL3577854)
Affinity DataKd:  2.50E+4nMAssay Description:Binding affinity to human full length PRMT5-MEP50 complex by Surface plasmon resonance methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50089221(CHEMBL3577854)
Affinity DataKd:  3.70E+4nMAssay Description:Binding affinity to human full length PRMT7 by Surface plasmon resonance methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50089221(CHEMBL3577854)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human full length PRMT7 expressed in Sf9 cells assessed as inhibition of H2B[23-37] methylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50396023(CHEMBL2169919)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of human full length PRMT7 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50089221(CHEMBL3577854)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human full length PRMT5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | S-[1-(adenin-9-yl)-1,5-dideoxy-beta-D-rib...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human full length PRMT5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50089221(CHEMBL3577854)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human full length PRMT7 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | S-[1-(adenin-9-yl)-1,5-dideoxy-beta-D-rib...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human full length PRMT7 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2016
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50089221(CHEMBL3577854)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human full length DNMT3A expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2016
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | S-[1-(adenin-9-yl)-1,5-dideoxy-beta-D-rib...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human full length DNMT3A expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2016
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3B(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50089221(CHEMBL3577854)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human full length DNMT3B expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2016
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3B(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | S-[1-(adenin-9-yl)-1,5-dideoxy-beta-D-rib...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human full length DNMT3B expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2016
Entry Details Article
PubMed