Compile Data Set for Download or QSAR
Report error Found 209 Enz. Inhib. hit(s) with all data for entry = 50046151
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096400(CHEMBL3577182)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096400(CHEMBL3577182)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096458(CHEMBL3577179)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096458(CHEMBL3577179)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096359(CHEMBL3577171)
Affinity DataEC50:  2nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096359(CHEMBL3577171)
Affinity DataEC50:  2nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096360(CHEMBL3577174)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096360(CHEMBL3577174)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096358(CHEMBL3577170)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096358(CHEMBL3577170)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096503(CHEMBL3577262)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096503(CHEMBL3577262)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096362(CHEMBL3577178)
Affinity DataEC50:  3.70nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096362(CHEMBL3577178)
Affinity DataEC50:  3.70nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096441(CHEMBL3577172)
Affinity DataEC50:  12nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096441(CHEMBL3577172)
Affinity DataEC50:  12nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096361(CHEMBL3577175)
Affinity DataEC50:  13nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096361(CHEMBL3577175)
Affinity DataEC50:  13nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 174(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096441(CHEMBL3577172)
Affinity DataEC50:  18nMAssay Description:Agonist activity at GPR174 (unknown origin) transfected in HEK293FT cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 174(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096441(CHEMBL3577172)
Affinity DataEC50:  18nMAssay Description:Agonist activity at GPR174 (unknown origin) transfected in HEK293FT cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096426(CHEMBL3577150)
Affinity DataEC50:  21nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096426(CHEMBL3577150)
Affinity DataEC50:  21nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 174(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096361(CHEMBL3577175)
Affinity DataEC50:  25nMAssay Description:Agonist activity at GPR174 (unknown origin) transfected in HEK293FT cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096422(CHEMBL3577137)
Affinity DataEC50:  25nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096422(CHEMBL3577137)
Affinity DataEC50:  25nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 174(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096361(CHEMBL3577175)
Affinity DataEC50:  25nMAssay Description:Agonist activity at GPR174 (unknown origin) transfected in HEK293FT cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096353(CHEMBL3577145)
Affinity DataEC50:  26nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096353(CHEMBL3577145)
Affinity DataEC50:  26nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  28nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  28nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 174(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096586(CHEMBL3577265)
Affinity DataEC50:  31nMAssay Description:Agonist activity at GPR174 (unknown origin) transfected in HEK293FT cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 174(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096586(CHEMBL3577265)
Affinity DataEC50:  31nMAssay Description:Agonist activity at GPR174 (unknown origin) transfected in HEK293FT cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096478(CHEMBL3577180)
Affinity DataEC50:  32nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096478(CHEMBL3577180)
Affinity DataEC50:  33nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 174(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096360(CHEMBL3577174)
Affinity DataEC50:  33nMAssay Description:Agonist activity at GPR174 (unknown origin) transfected in HEK293FT cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 174(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096360(CHEMBL3577174)
Affinity DataEC50:  33nMAssay Description:Agonist activity at GPR174 (unknown origin) transfected in HEK293FT cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096350(CHEMBL3577138)
Affinity DataEC50:  39nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096350(CHEMBL3577138)
Affinity DataEC50:  39nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 174(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096583(CHEMBL3577263)
Affinity DataEC50:  40nMAssay Description:Agonist activity at GPR174 (unknown origin) transfected in HEK293FT cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 174(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096583(CHEMBL3577263)
Affinity DataEC50:  40nMAssay Description:Agonist activity at GPR174 (unknown origin) transfected in HEK293FT cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 174(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096359(CHEMBL3577171)
Affinity DataEC50:  44nMAssay Description:Agonist activity at GPR174 (unknown origin) transfected in HEK293FT cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 174(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096359(CHEMBL3577171)
Affinity DataEC50:  44nMAssay Description:Agonist activity at GPR174 (unknown origin) transfected in HEK293FT cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096357(CHEMBL3577151)
Affinity DataEC50:  45nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096357(CHEMBL3577151)
Affinity DataEC50:  45nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096443(CHEMBL3577176)
Affinity DataEC50:  53nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096443(CHEMBL3577176)
Affinity DataEC50:  54nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096502(CHEMBL3577181)
Affinity DataEC50:  55nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096502(CHEMBL3577181)
Affinity DataEC50:  56nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096355(CHEMBL3577149)
Affinity DataEC50:  58nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096351(CHEMBL3577140)
Affinity DataEC50:  58nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
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