Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50046021
TargetAlpha-1A adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091350(CHEMBL3582270)
Affinity DataIC50: 0.600nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1A adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM31046(SMR000059054 | cid_91430 | 3-[4,5-dihydro-1H-imida...)
Affinity DataIC50: 1.10nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1A adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091350(CHEMBL3582270)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1B adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091350(CHEMBL3582270)
Affinity DataIC50: 2.20nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1D adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091351(CHEMBL3582269)
Affinity DataIC50: 2.5nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1A adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091352(CHEMBL3582268)
Affinity DataIC50: 3.90nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1A adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091352(CHEMBL3582268)
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1B adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091351(CHEMBL3582269)
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1B adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091351(CHEMBL3582269)
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1D adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091352(CHEMBL3582268)
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1D adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091349(CHEMBL3582271)
Affinity DataIC50: 8.80nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1A adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM31046(SMR000059054 | cid_91430 | 3-[4,5-dihydro-1H-imida...)
Affinity DataIC50: 11nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1B adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM31046(SMR000059054 | cid_91430 | 3-[4,5-dihydro-1H-imida...)
Affinity DataIC50: 13nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1D adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091349(CHEMBL3582271)
Affinity DataIC50: 16nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1B adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091349(CHEMBL3582271)
Affinity DataIC50: 34nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1D adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091348(CHEMBL3582272)
Affinity DataIC50: 45nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1D adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091348(CHEMBL3582272)
Affinity DataIC50: 52nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1A adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091348(CHEMBL3582272)
Affinity DataIC50: 52nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1B adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091350(CHEMBL3582270)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1B adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091350(CHEMBL3582270)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1A adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091350(CHEMBL3582270)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1D adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM31046(SMR000059054 | cid_91430 | 3-[4,5-dihydro-1H-imida...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1A adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091351(CHEMBL3582269)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1A adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091352(CHEMBL3582268)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1A adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091349(CHEMBL3582271)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1A adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM31046(SMR000059054 | cid_91430 | 3-[4,5-dihydro-1H-imida...)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1B adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091349(CHEMBL3582271)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1B adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM31046(SMR000059054 | cid_91430 | 3-[4,5-dihydro-1H-imida...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1D adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091349(CHEMBL3582271)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1D adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091348(CHEMBL3582272)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1D adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091348(CHEMBL3582272)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1B adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091348(CHEMBL3582272)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1A adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2016
Entry Details Article
PubMed