Compile Data Set for Download or QSAR
Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 50046161
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097128(CHEMBL3580976)
Affinity DataIC50: 85nMAssay Description:Inhibition of PAK1 in human EBC1 cells assessed as inhibition of MEK phosphorylation at S298 after 2 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50096231(CHEMBL3580975)
Affinity DataIC50: 110nMAssay Description:Inhibition of PAK1 in human EBC1 cells assessed as inhibition of MEK phosphorylation at S298 after 2 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097133(CHEMBL3580968)
Affinity DataIC50: 120nMAssay Description:Inhibition of PAK1 in human EBC1 cells assessed as inhibition of MEK phosphorylation at S298 after 2 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097134(CHEMBL3580972)
Affinity DataIC50: 281nMAssay Description:Inhibition of PAK1 in human EBC1 cells assessed as inhibition of MEK phosphorylation at S298 after 2 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097135(CHEMBL3580974)
Affinity DataIC50: 362nMAssay Description:Inhibition of PAK1 in human EBC1 cells assessed as inhibition of MEK phosphorylation at S298 after 2 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097132(CHEMBL3580962)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of PAK1 in human EBC1 cells assessed as inhibition of MEK phosphorylation at S298 after 2 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097131(CHEMBL3580667)
Affinity DataKi:  2nMAssay Description:Inhibition of human PAK4More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097144(CHEMBL3580963)
Affinity DataKi:  4nMAssay Description:Inhibition of human recombinant PAK4 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50096231(CHEMBL3580975)
Affinity DataKi:  4nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097128(CHEMBL3580976)
Affinity DataKi:  5nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097135(CHEMBL3580974)
Affinity DataKi:  5nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097128(CHEMBL3580976)
Affinity DataKi:  5.30nMAssay Description:Inhibition of aurora A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097127(CHEMBL3580949)
Affinity DataKi:  12nMAssay Description:Inhibition of human recombinant PAK4 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097134(CHEMBL3580972)
Affinity DataKi:  12nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM101618(US8530652, 114)
Affinity DataKi:  15nMAssay Description:Inhibition of N-terminal His6-tagged human recombinant PAK4 (300 to 591 amino acids) using peptide-7 substrate by pyruvate kinase and lactate dehydro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097121(CHEMBL3580954)
Affinity DataKi:  18nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097144(CHEMBL3580963)
Affinity DataKi:  21nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097127(CHEMBL3580949)
Affinity DataKi:  22nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097132(CHEMBL3580962)
Affinity DataKi:  26nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097140(CHEMBL3580967)
Affinity DataKi:  27nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097133(CHEMBL3580968)
Affinity DataKi:  31nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097122(CHEMBL3580953)
Affinity DataKi:  33nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097124(CHEMBL3580951)
Affinity DataKi:  33nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097132(CHEMBL3580962)
Affinity DataKi:  38nMAssay Description:Inhibition of human recombinant PAK4 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM101618(US8530652, 114)
Affinity DataKi:  39nMAssay Description:Inhibition of PAK1 (unknown origin) using Syntide2 peptide substrate by pyruvate kinase and lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase PAK 4(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097133(CHEMBL3580968)
Affinity DataKi:  42nMAssay Description:Inhibition of human recombinant PAK4 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097119(CHEMBL3580956)
Affinity DataKi:  45nMAssay Description:Inhibition of human recombinant PAK4 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097123(CHEMBL3580952)
Affinity DataKi:  48nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097130(CHEMBL3580948)
Affinity DataKi:  49nMAssay Description:Inhibition of human PAK4More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097131(CHEMBL3580667)
Affinity DataKi:  50nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097146(CHEMBL3580960)
Affinity DataKi:  80nMAssay Description:Inhibition of human recombinant PAK4 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097130(CHEMBL3580948)
Affinity DataKi:  100nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097145(CHEMBL3580961)
Affinity DataKi:  100nMAssay Description:Inhibition of human recombinant PAK4 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097134(CHEMBL3580972)
Affinity DataKi:  106nMAssay Description:Inhibition of human recombinant PAK4 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097139(CHEMBL3580969)
Affinity DataKi:  117nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097119(CHEMBL3580956)
Affinity DataKi:  119nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097143(CHEMBL3580964)
Affinity DataKi:  138nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097140(CHEMBL3580967)
Affinity DataKi:  144nMAssay Description:Inhibition of human recombinant PAK4 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097145(CHEMBL3580961)
Affinity DataKi:  157nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097126(CHEMBL3580950)
Affinity DataKi:  179nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097136(CHEMBL3580973)
Affinity DataKi:  179nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097146(CHEMBL3580960)
Affinity DataKi:  245nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50096231(CHEMBL3580975)
Affinity DataKi:  272nMAssay Description:Inhibition of human recombinant PAK4 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097149(CHEMBL3580957)
Affinity DataKi:  283nMAssay Description:Inhibition of human recombinant PAK4 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097142(CHEMBL3580965)
Affinity DataKi:  346nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097149(CHEMBL3580957)
Affinity DataKi:  454nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097135(CHEMBL3580974)
Affinity DataKi:  455nMAssay Description:Inhibition of human recombinant PAK4 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097128(CHEMBL3580976)
Affinity DataKi:  547nMAssay Description:Inhibition of human recombinant PAK4 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097148(CHEMBL3580958)
Affinity DataKi:  561nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Shanghai Chempartner

Curated by ChEMBL
LigandPNGBDBM50097143(CHEMBL3580964)
Affinity DataKi:  563nMAssay Description:Inhibition of human recombinant PAK4 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
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