Compile Data Set for Download or QSAR
Report error Found 57 Enz. Inhib. hit(s) with all data for entry = 50046370
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108676(CHEMBL3596502)
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of [35S]MK499 binding to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108650(CHEMBL3596509)
Affinity DataIC50: 2.18E+3nMAssay Description:Inhibition of [35S]MK499 binding to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108672(CHEMBL3596506)
Affinity DataIC50: 1.69E+4nMAssay Description:Inhibition of [35S]MK499 binding to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108681(CHEMBL3596516)
Affinity DataIC50: 1.79E+4nMAssay Description:Inhibition of [35S]MK499 binding to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108684(CHEMBL3596513)
Affinity DataIC50: 2.08E+4nMAssay Description:Inhibition of [35S]MK499 binding to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108647(CHEMBL3596512)
Affinity DataIC50: 2.11E+4nMAssay Description:Inhibition of [35S]MK499 binding to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108673(CHEMBL3596505)
Affinity DataIC50: 2.19E+4nMAssay Description:Inhibition of [35S]MK499 binding to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108651(CHEMBL3596508)
Affinity DataIC50: 2.23E+4nMAssay Description:Inhibition of [35S]MK499 binding to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108674(CHEMBL3596504)
Affinity DataIC50: 2.38E+4nMAssay Description:Inhibition of [35S]MK499 binding to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108679(CHEMBL3596518)
Affinity DataIC50: 2.43E+4nMAssay Description:Inhibition of [35S]MK499 binding to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108671(CHEMBL3596507)
Affinity DataIC50: 2.55E+4nMAssay Description:Inhibition of [35S]MK499 binding to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108678(CHEMBL3596589)
Affinity DataIC50: 3.92E+4nMAssay Description:Inhibition of [35S]MK499 binding to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108682(CHEMBL3596515)
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of [35S]MK499 binding to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108648(CHEMBL3596511)
Affinity DataIC50: 4.76E+4nMAssay Description:Inhibition of [35S]MK499 binding to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108675(CHEMBL3596503)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of [35S]MK499 binding to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108680(CHEMBL3596517)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of [35S]MK499 binding to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108683(CHEMBL3596514)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of [35S]MK499 binding to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108677(CHEMBL3596590)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of [35S]MK499 binding to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108649(CHEMBL3596510)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of [35S]MK499 binding to human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108680(CHEMBL3596517)
Affinity DataKi:  1.40nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108684(CHEMBL3596513)
Affinity DataKi:  4.80nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108679(CHEMBL3596518)
Affinity DataKi:  5.20nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108674(CHEMBL3596504)
Affinity DataKi:  5.30nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108676(CHEMBL3596502)
Affinity DataKi:  5.5nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108681(CHEMBL3596516)
Affinity DataKi:  6.70nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108647(CHEMBL3596512)
Affinity DataKi:  7.70nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108675(CHEMBL3596503)
Affinity DataKi:  8.60nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108648(CHEMBL3596511)
Affinity DataKi:  8.90nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108677(CHEMBL3596590)
Affinity DataKi:  9.40nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108672(CHEMBL3596506)
Affinity DataKi:  10nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108673(CHEMBL3596505)
Affinity DataKi:  13nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108678(CHEMBL3596589)
Affinity DataKi:  20nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108682(CHEMBL3596515)
Affinity DataKi:  23nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108683(CHEMBL3596514)
Affinity DataKi:  25nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108649(CHEMBL3596510)
Affinity DataKi:  27nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108671(CHEMBL3596507)
Affinity DataKi:  38nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108651(CHEMBL3596508)
Affinity DataKi:  40nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108650(CHEMBL3596509)
Affinity DataKi:  93nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108672(CHEMBL3596506)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108679(CHEMBL3596518)
Affinity DataKi:  1.26E+3nMAssay Description:Inhibition of human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108674(CHEMBL3596504)
Affinity DataKi:  1.37E+3nMAssay Description:Inhibition of human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108676(CHEMBL3596502)
Affinity DataKi:  1.45E+3nMAssay Description:Inhibition of human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108649(CHEMBL3596510)
Affinity DataKi:  1.55E+3nMAssay Description:Inhibition of human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108680(CHEMBL3596517)
Affinity DataKi:  1.92E+3nMAssay Description:Inhibition of human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108684(CHEMBL3596513)
Affinity DataKi:  2.41E+3nMAssay Description:Inhibition of human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108673(CHEMBL3596505)
Affinity DataKi:  2.72E+3nMAssay Description:Inhibition of human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108671(CHEMBL3596507)
Affinity DataKi:  3.09E+3nMAssay Description:Inhibition of human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108675(CHEMBL3596503)
Affinity DataKi:  3.55E+3nMAssay Description:Inhibition of human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108681(CHEMBL3596516)
Affinity DataKi:  4.29E+3nMAssay Description:Inhibition of human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108647(CHEMBL3596512)
Affinity DataKi:  4.99E+3nMAssay Description:Inhibition of human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
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