Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50046339
TargetProstaglandin G/H synthase 2(Human)
Technische Universitat Dresden

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 130nMAssay Description:Inhibition of recombinant human COX-2 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2016
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Technische Universitat Dresden

Curated by ChEMBL
LigandPNGBDBM50106762(CHEMBL3601277)
Affinity DataIC50: 220nMAssay Description:Inhibition of recombinant human COX-2 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2016
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Technische Universitat Dresden

Curated by ChEMBL
LigandPNGBDBM50106760(CHEMBL3601279)
Affinity DataIC50: 280nMAssay Description:Inhibition of recombinant human COX-2 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2016
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Technische Universitat Dresden

Curated by ChEMBL
LigandPNGBDBM50106763(CHEMBL3601276)
Affinity DataIC50: 890nMAssay Description:Inhibition of recombinant human COX-2 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2016
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Technische Universitat Dresden

Curated by ChEMBL
LigandPNGBDBM50106761(CHEMBL3601278)
Affinity DataIC50: 970nMAssay Description:Inhibition of recombinant human COX-2 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2016
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Technische Universitat Dresden

Curated by ChEMBL
LigandPNGBDBM50428519(CHEMBL2336619)
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of recombinant human COX-2 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2016
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Technische Universitat Dresden

Curated by ChEMBL
LigandPNGBDBM50106759(CHEMBL3601280)
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of recombinant human COX-2 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2016
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Technische Universitat Dresden

Curated by ChEMBL
LigandPNGBDBM50106760(CHEMBL3601279)
Affinity DataIC50: 6.10E+4nMAssay Description:Inhibition of ovine COX-1 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazine to resoru...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2016
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Technische Universitat Dresden

Curated by ChEMBL
LigandPNGBDBM50106759(CHEMBL3601280)
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibition of ovine COX-1 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazine to resoru...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2016
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Technische Universitat Dresden

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of ovine COX-1 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazine to resoru...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2016
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Technische Universitat Dresden

Curated by ChEMBL
LigandPNGBDBM50106761(CHEMBL3601278)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of ovine COX-1 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazine to resoru...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2016
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Technische Universitat Dresden

Curated by ChEMBL
LigandPNGBDBM50106762(CHEMBL3601277)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of ovine COX-1 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazine to resoru...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2016
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Technische Universitat Dresden

Curated by ChEMBL
LigandPNGBDBM50106763(CHEMBL3601276)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of ovine COX-1 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazine to resoru...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2016
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Technische Universitat Dresden

Curated by ChEMBL
LigandPNGBDBM50428519(CHEMBL2336619)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of ovine COX-1 assessed as reduction of prostaglandin-G2 to prostaglandin-H2 and oxidation of 10-acetyl-3,7-dihydroxyphenoxazine to resoru...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2016
Entry Details Article
PubMed