Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50046497
TargetCoagulation factor X(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50115828(CHEMBL3612132)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of human F10a using S-2765 as substrate preincubated for 10 mins followed by substrate addition by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM7840(RIVAROXABAN | US8822458, 97 | US8822458, 44)
Affinity DataIC50: 14nMAssay Description:Inhibition of human F10a using S-2765 as substrate preincubated for 10 mins followed by substrate addition by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50115823(CHEMBL3612128)
Affinity DataIC50: 16nMAssay Description:Inhibition of human F10a using S-2765 as substrate preincubated for 10 mins followed by substrate addition by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50115827(CHEMBL3612122)
Affinity DataIC50: 17nMAssay Description:Inhibition of human F10a using S-2765 as substrate preincubated for 10 mins followed by substrate addition by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50115824(CHEMBL3612126)
Affinity DataIC50: 26nMAssay Description:Inhibition of human F10a using S-2765 as substrate preincubated for 10 mins followed by substrate addition by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50115826(CHEMBL3612123)
Affinity DataIC50: 29nMAssay Description:Inhibition of human F10a using S-2765 as substrate preincubated for 10 mins followed by substrate addition by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2016
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50115827(CHEMBL3612122)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of bovine plasma thrombin using S-2238 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2016
Entry Details Article
PubMed
TargetTrypsin(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50115827(CHEMBL3612122)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of trypsin (unknown origin) using S-2222 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2016
Entry Details Article
PubMed