Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50046475
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114404(CHEMBL3608325)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114409(CHEMBL3609809)
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114408(CHEMBL3609810)
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114400(CHEMBL3608329)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114409(CHEMBL3609809)
Affinity DataKi:  3.90E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as disappearance of NADH fluorescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114401(CHEMBL3608328)
Affinity DataIC50: 4.10E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114403(CHEMBL3608326)
Affinity DataIC50: 4.10E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114409(CHEMBL3609809)
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114407(CHEMBL3197264)
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114402(CHEMBL3608327)
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114409(CHEMBL3609809)
Affinity DataKi:  4.70E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using NADH as substrate assessed as disappearance of NADH fluorescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114399(CHEMBL3608330)
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114404(CHEMBL3608325)
Affinity DataIC50: 5.20E+4nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114400(CHEMBL3608329)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114403(CHEMBL3608326)
Affinity DataIC50: 1.05E+5nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114399(CHEMBL3608330)
Affinity DataIC50: 1.15E+5nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114405(CHEMBL3609813)
Affinity DataIC50: 1.25E+5nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114405(CHEMBL3609813)
Affinity DataIC50: 1.34E+5nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114407(CHEMBL3197264)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114406(CHEMBL3609811)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114408(CHEMBL3609810)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114411(CHEMBL3608331)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114410(CHEMBL3608332)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114401(CHEMBL3608328)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114412(CHEMBL3609812)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human liver purified lactate dehydrogenase-A using pyruvate as substrate assessed as NADH oxidation for 3 mins by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50114402(CHEMBL3608327)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of lactate dehydrogenase-A in human Raji cells assessed as reduction of intracellular lactate level after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed