Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50047158
TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50148552(CHEMBL3770150)
Affinity DataKd:  770nMAssay Description:Competitive binding affinity to partial length human CREBBP expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50150909(CHEMBL3774461)
Affinity DataIC50: 1.50E+3nMAssay Description:Binding affinity to N-terminal GST-tagged recombinant human CREBBP expressed in Escherichia coli after 2 hrs using BET bromodomain ligand by TR-FRET ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2017
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50150909(CHEMBL3774461)
Affinity DataKd:  4.20E+3nMAssay Description:Competitive binding affinity to partial length human CREBBP expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2017
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50443249(Ischemin)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of CREBBP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2017
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50150939(CHEMBL3775960)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity to CREBBP (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2017
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50150919(CHEMBL3775048)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to N-terminal GST-tagged recombinant human CREBBP expressed in Escherichia coli after 2 hrs using BET bromodomain ligand by TR-FRET ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2017
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50150938(CHEMBL3775724)
Affinity DataKd:  1.30E+4nMAssay Description:Competitive binding affinity to partial length human CREBBP expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2017
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50148550(CHEMBL3770132)
Affinity DataKd:  2.90E+4nMAssay Description:Competitive binding affinity to partial length human CREBBP expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2017
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50150938(CHEMBL3775724)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity to N-terminal GST-tagged recombinant human CREBBP expressed in Escherichia coli after 2 hrs using BET bromodomain ligand by TR-FRET ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2017
Entry Details Article
PubMed