Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 50046192
LigandPNGBDBM50098596(CHEMBL3594313)
Affinity DataKi:  0.700nMAssay Description:Inhibition of human recombinant TF/F7a complex using S2288 as substrate preincubated for 15 mins followed by protein addition measured for 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
LigandPNGBDBM50098595(CHEMBL3594314)
Affinity DataKi:  1.60nMAssay Description:Inhibition of human recombinant TF/F7a complex using S2288 as substrate preincubated for 15 mins followed by protein addition measured for 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
LigandPNGBDBM50098598(CHEMBL3594311)
Affinity DataKi:  5.20nMAssay Description:Inhibition of human recombinant TF/F7a complex using S2288 as substrate preincubated for 15 mins followed by protein addition measured for 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
LigandPNGBDBM50098600(CHEMBL3594315)
Affinity DataKi:  8nMAssay Description:Inhibition of human recombinant TF/F7a complex using S2288 as substrate preincubated for 15 mins followed by protein addition measured for 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50098599(CHEMBL3594310)
Affinity DataKi:  8nMAssay Description:Inhibition of human recombinant TF/F7a complex using S2288 as substrate preincubated for 15 mins followed by protein addition measured for 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetKallikrein-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098591(CHEMBL3594305)
Affinity DataKi:  18nMAssay Description:Inhibition of human tissue kallikrein 1 measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetKallikrein-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098597(CHEMBL3594312)
Affinity DataKi:  22nMAssay Description:Inhibition of human tissue kallikrein 1 measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
LigandPNGBDBM50098597(CHEMBL3594312)
Affinity DataKi:  30nMAssay Description:Inhibition of human recombinant TF/F7a complex using S2288 as substrate preincubated for 15 mins followed by protein addition measured for 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098596(CHEMBL3594313)
Affinity DataKi:  41nMAssay Description:Inhibition of human APC measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098596(CHEMBL3594313)
Affinity DataKi:  50nMAssay Description:Inhibition of human plasma kallikrein using S2302 as substrate measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetTrypsin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098596(CHEMBL3594313)
Affinity DataKi:  58nMAssay Description:Inhibition of human trypsin measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetKallikrein-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098595(CHEMBL3594314)
Affinity DataKi:  100nMAssay Description:Inhibition of human tissue kallikrein 1 measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetKallikrein-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098599(CHEMBL3594310)
Affinity DataKi:  100nMAssay Description:Inhibition of human tissue kallikrein 1 measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetKallikrein-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098598(CHEMBL3594311)
Affinity DataKi:  100nMAssay Description:Inhibition of human tissue kallikrein 1 measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098596(CHEMBL3594313)
Affinity DataKi:  180nMAssay Description:Inhibition of human thrombin using S2238 as substrate measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
LigandPNGBDBM50098591(CHEMBL3594305)
Affinity DataKi:  400nMAssay Description:Inhibition of human recombinant TF/F7a complex using S2288 as substrate preincubated for 15 mins followed by protein addition measured for 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetVitamin K-dependent protein C(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098595(CHEMBL3594314)
Affinity DataKi:  830nMAssay Description:Inhibition of human APC measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
LigandPNGBDBM50098592(CHEMBL3594304)
Affinity DataKi:  920nMAssay Description:Inhibition of human recombinant TF/F7a complex using S2288 as substrate preincubated for 15 mins followed by protein addition measured for 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098595(CHEMBL3594314)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of human F10a using S2222 as substrate measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098599(CHEMBL3594310)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of human APC measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098595(CHEMBL3594314)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of human plasma kallikrein using S2302 as substrate measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098598(CHEMBL3594311)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of human APC measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetKallikrein-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098596(CHEMBL3594313)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of human tissue kallikrein 1 measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetTrypsin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098595(CHEMBL3594314)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of human trypsin measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098591(CHEMBL3594305)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibition of human APC measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetTrypsin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098598(CHEMBL3594311)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of human trypsin measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098599(CHEMBL3594310)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of human F10a using S2222 as substrate measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098598(CHEMBL3594311)
Affinity DataKi:  3.30E+3nMAssay Description:Inhibition of human F10a using S2222 as substrate measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetTrypsin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098599(CHEMBL3594310)
Affinity DataKi:  3.60E+3nMAssay Description:Inhibition of human trypsin measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098598(CHEMBL3594311)
Affinity DataKi:  3.60E+3nMAssay Description:Inhibition of human plasma kallikrein using S2302 as substrate measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098598(CHEMBL3594311)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of human thrombin using S2238 as substrate measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098599(CHEMBL3594310)
Affinity DataKi:  4.60E+3nMAssay Description:Inhibition of human plasma kallikrein using S2302 as substrate measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
LigandPNGBDBM50098666(CHEMBL3594307)
Affinity DataKi:  4.60E+3nMAssay Description:Inhibition of human recombinant TF/F7a complex using S2288 as substrate preincubated for 15 mins followed by protein addition measured for 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
LigandPNGBDBM50098594(CHEMBL3594302)
Affinity DataKi:  4.60E+3nMAssay Description:Inhibition of human recombinant TF/F7a complex using S2288 as substrate preincubated for 15 mins followed by protein addition measured for 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098597(CHEMBL3594312)
Affinity DataKi:  4.80E+3nMAssay Description:Inhibition of human F10a using S2222 as substrate measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098596(CHEMBL3594313)
Affinity DataKi:  5.50E+3nMAssay Description:Inhibition of human F10a using S2222 as substrate measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098599(CHEMBL3594310)
Affinity DataKi:  5.80E+3nMAssay Description:Inhibition of human thrombin using S2238 as substrate measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098591(CHEMBL3594305)
Affinity DataKi: >6.00E+3nMAssay Description:Inhibition of human plasma kallikrein using S2302 as substrate measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098597(CHEMBL3594312)
Affinity DataKi: >6.00E+3nMAssay Description:Inhibition of human plasma kallikrein using S2302 as substrate measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetTrypsin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098597(CHEMBL3594312)
Affinity DataKi: >6.00E+3nMAssay Description:Inhibition of human trypsin measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetTrypsin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098591(CHEMBL3594305)
Affinity DataKi: >6.00E+3nMAssay Description:Inhibition of human trypsin measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
LigandPNGBDBM50098593(CHEMBL3594303)
Affinity DataKi:  6.10E+3nMAssay Description:Inhibition of human recombinant TF/F7a complex using S2288 as substrate preincubated for 15 mins followed by protein addition measured for 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098595(CHEMBL3594314)
Affinity DataKi:  6.70E+3nMAssay Description:Inhibition of human thrombin using S2238 as substrate measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098591(CHEMBL3594305)
Affinity DataKi: >9.00E+3nMAssay Description:Inhibition of human F10a using S2222 as substrate measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
LigandPNGBDBM50098601(CHEMBL3594309)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of human recombinant TF/F7a complex using S2288 as substrate preincubated for 15 mins followed by protein addition measured for 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098597(CHEMBL3594312)
Affinity DataKi: >1.30E+4nMAssay Description:Inhibition of human thrombin using S2238 as substrate measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098591(CHEMBL3594305)
Affinity DataKi: >1.30E+4nMAssay Description:Inhibition of human thrombin using S2238 as substrate measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098597(CHEMBL3594312)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibition of human APC measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50098595(CHEMBL3594314)
Affinity DataKi:  1.60E+4nMAssay Description:Inhibition of human F9a measured for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
LigandPNGBDBM50098708(CHEMBL3594306)
Affinity DataKi: >1.80E+4nMAssay Description:Inhibition of human recombinant TF/F7a complex using S2288 as substrate preincubated for 15 mins followed by protein addition measured for 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2016
Entry Details Article
PubMed
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