Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50046439
TargetBaculoviral IAP repeat-containing protein 3(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandPNGBDBM50112346(CHEMBL3609325)
Affinity DataIC50: 3nMAssay Description:Inhibition of cIAP BIR2-3 domain (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandPNGBDBM50112346(CHEMBL3609325)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of XIAP BIR3 domain (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandPNGBDBM50112346(CHEMBL3609325)
Affinity DataEC50:  9.40nMAssay Description:Inhibition of XIAP (unknown origin) by caspase-3 rescue assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandPNGBDBM50112346(CHEMBL3609325)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetCytochrome P450 2B6(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandPNGBDBM50112346(CHEMBL3609325)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human CYP2B6More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C8(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandPNGBDBM50112346(CHEMBL3609325)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human CYP2C8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandPNGBDBM50112346(CHEMBL3609325)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandPNGBDBM50112346(CHEMBL3609325)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandPNGBDBM50112346(CHEMBL3609325)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human CYP2D6More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandPNGBDBM50112346(CHEMBL3609325)
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of PXR (unknown origin) by receptor transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed