Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50046473
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50114377(CHEMBL3604283)
Affinity DataIC50: 11nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50114376(CHEMBL3604335)
Affinity DataIC50: 12nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50114375(CHEMBL3604336)
Affinity DataIC50: 15nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50114382(CHEMBL3604349)
Affinity DataIC50: 16nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50114374(CHEMBL3604337)
Affinity DataIC50: 94nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50114381(CHEMBL3604348)
Affinity DataIC50: 100nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50116355(CHEMBL3604344)
Affinity DataIC50: 190nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM10404(galantamine | (1S,12S,14R)-9-methoxy-4-methyl-11-o...)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM10404(galantamine | (1S,12S,14R)-9-methoxy-4-methyl-11-o...)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50114380(CHEMBL3604347)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50237933(N-(14-methylallyl)norgalanthamine | CHEMBL442287)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50114389(CHEMBL3604356)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50114390(CHEMBL3604357)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50114384(CHEMBL3604351)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50114386(CHEMBL3604353)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50114385(CHEMBL3604352)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50114379(CHEMBL3604346)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50114387(CHEMBL3604354)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50116350(CHEMBL3604341)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50114383(CHEMBL3604350)
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50114378(CHEMBL3604345)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50116352(CHEMBL3604339)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50116356(CHEMBL3604343)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50114388(CHEMBL3604355)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50116351(CHEMBL3604342)
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50114391(CHEMBL3604358)
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50116354(CHEMBL3604338)
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Medical University of Sofia

Curated by ChEMBL
LigandPNGBDBM50116353(CHEMBL3604340)
Affinity DataIC50: 8.40E+4nMAssay Description:Inhibition of Torpedo californica AChE using ATCI substrate incubated for 30 mins by Ellman's method based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2016
Entry Details Article
PubMed