Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50046548
TargetVascular endothelial growth factor receptor 2(Human)
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 6nMAssay Description:Inhibition of VEGFR2 (unknown origin) using Tyr1 peptide as substrate after 1 hr by FRET-based assay in presence of 10 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50118114(CHEMBL3612230)
Affinity DataIC50: 10nMAssay Description:Inhibition of VEGFR2 (unknown origin) using Tyr1 peptide as substrate after 1 hr by FRET-based assay in presence of 10 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50118116(CHEMBL3612232)
Affinity DataIC50: 11nMAssay Description:Inhibition of VEGFR2 (unknown origin) using Tyr1 peptide as substrate after 1 hr by FRET-based assay in presence of 10 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50118117(CHEMBL3612233)
Affinity DataIC50: 15nMAssay Description:Inhibition of VEGFR2 (unknown origin) using Tyr1 peptide as substrate after 1 hr by FRET-based assay in presence of 10 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50118118(CHEMBL3612234)
Affinity DataIC50: 16nMAssay Description:Inhibition of VEGFR2 (unknown origin) using Tyr1 peptide as substrate after 1 hr by FRET-based assay in presence of 10 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50118115(CHEMBL3612231)
Affinity DataIC50: 28nMAssay Description:Inhibition of VEGFR2 (unknown origin) using Tyr1 peptide as substrate after 1 hr by FRET-based assay in presence of 10 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataIC50: 90nMAssay Description:Inhibition of human VEGFR2 after 1.5 to 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetVascular endothelial growth factor receptor 2(Human)
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50118127(CHEMBL3612227)
Affinity DataIC50: 94nMAssay Description:Inhibition of VEGFR2 (unknown origin) using Tyr1 peptide as substrate after 1 hr by FRET-based assay in presence of 10 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50118128(CHEMBL3612228)
Affinity DataIC50: 107nMAssay Description:Inhibition of VEGFR2 (unknown origin) using Tyr1 peptide as substrate after 1 hr by FRET-based assay in presence of 10 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50118113(CHEMBL3612229)
Affinity DataIC50: 206nMAssay Description:Inhibition of VEGFR2 (unknown origin) using Tyr1 peptide as substrate after 1 hr by FRET-based assay in presence of 10 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50118122(CHEMBL3612325)
Affinity DataIC50: 988nMAssay Description:Inhibition of VEGFR2 (unknown origin) using Tyr1 peptide as substrate after 1 hr by FRET-based assay in presence of 10 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50118119(CHEMBL3612235)
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibition of VEGFR2 (unknown origin) using Tyr1 peptide as substrate after 1 hr by FRET-based assay in presence of 10 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50118120(CHEMBL3612323)
Affinity DataIC50: 1.39E+3nMAssay Description:Inhibition of VEGFR2 (unknown origin) using Tyr1 peptide as substrate after 1 hr by FRET-based assay in presence of 10 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50118123(CHEMBL3612326)
Affinity DataIC50: 1.95E+3nMAssay Description:Inhibition of VEGFR2 (unknown origin) using Tyr1 peptide as substrate after 1 hr by FRET-based assay in presence of 10 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50118121(CHEMBL3612324)
Affinity DataIC50: 8.36E+3nMAssay Description:Inhibition of VEGFR2 (unknown origin) using Tyr1 peptide as substrate after 1 hr by FRET-based assay in presence of 10 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50118124(CHEMBL3612224)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of VEGFR2 (unknown origin) using Tyr1 peptide as substrate after 1 hr by FRET-based assay in presence of 10 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50118125(CHEMBL3612225)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of VEGFR2 (unknown origin) using Tyr1 peptide as substrate after 1 hr by FRET-based assay in presence of 10 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50118126(CHEMBL3612226)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of VEGFR2 (unknown origin) using Tyr1 peptide as substrate after 1 hr by FRET-based assay in presence of 10 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed