Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50046769
TargetVascular endothelial growth factor receptor 2(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50130404(CHEMBL3633687)
Affinity DataIC50: 8nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM5875(N-[5-(ethanesulfonyl)-2-methoxyphenyl]-5-[3-(pyrid...)
Affinity DataIC50: 22nMAssay Description:Inhibition of GST-tagged human recombinant VEGFR2 kinase expressed in Sf9 insect cells by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataIC50: 39nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50130405(CHEMBL3633688)
Affinity DataIC50: 45nMAssay Description:Inhibition of His6-tagged KDR 789 to 1354 residues (unknown origin) using biotin-Ahx-AEEEYFFLA-amide substrate incubated for 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50130403(CHEMBL3633689)
Affinity DataIC50: 49nMAssay Description:Inhibition of GST-tagged human KDR expressed in Sf21 cells using 4:1 polyglutamic acid/tyrosine substrate incubated for 15 mins by scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50130408(CHEMBL3633692)
Affinity DataIC50: 6.96E+3nMAssay Description:Inhibition of GST-tagged human recombinant VEGFR2 kinase expressed in Sf9 insect cells by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50130410(CHEMBL3633690)
Affinity DataIC50: 4.01E+4nMAssay Description:Inhibition of GST-tagged human recombinant VEGFR2 kinase expressed in Sf9 insect cells by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50130406(CHEMBL3633696)
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of GST-tagged human recombinant VEGFR2 kinase expressed in Sf9 insect cells by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50130407(CHEMBL3633695)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of GST-tagged human recombinant VEGFR2 kinase expressed in Sf9 insect cells by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50130409(CHEMBL3633691)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of GST-tagged human recombinant VEGFR2 kinase expressed in Sf9 insect cells by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed