Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50046807
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50132143(CHEMBL3633720)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50132137(CHEMBL3633878)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131904(CHEMBL3633888)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131902(CHEMBL3633890)
Affinity DataEC50:  32nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131999(CHEMBL3633881)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131906(CHEMBL3633886)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131899(CHEMBL3633893)
Affinity DataEC50:  43nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131905(CHEMBL3633887)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131993(CHEMBL3633883)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131946(CHEMBL3633884)
Affinity DataEC50:  52nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131994(CHEMBL3633882)
Affinity DataEC50:  52nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50132000(CHEMBL3633880)
Affinity DataEC50:  54nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50132131(CHEMBL3633879)
Affinity DataEC50:  59nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131903(CHEMBL3633889)
Affinity DataEC50:  78nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50132141(CHEMBL3633721)
Affinity DataEC50:  118nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131931(CHEMBL3633885)
Affinity DataEC50:  193nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131897(CHEMBL3633894)
Affinity DataEC50:  670nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131896(CHEMBL3633895)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131895(CHEMBL3633896)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131901(CHEMBL3633891)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131900(CHEMBL3633892)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed