Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50006329
TargetPoly [ADP-ribose] polymerase tankyrase-1/tankyrase-2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50498904(CHEMBL3734991)
Affinity DataEC50:  2nMAssay Description:Inhibition of Tankyrase in human DLD1 cells assessed as T-cell factor level after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1/tankyrase-2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50498905(CHEMBL3736012)
Affinity DataEC50:  7nMAssay Description:Inhibition of Tankyrase in human DLD1 cells assessed as T-cell factor level after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1/tankyrase-2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50498903(CHEMBL3735964)
Affinity DataEC50:  31nMAssay Description:Inhibition of Tankyrase in human DLD1 cells assessed as T-cell factor level after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1/tankyrase-2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50498900(CHEMBL3736145)
Affinity DataEC50:  47nMAssay Description:Inhibition of Tankyrase in human DLD1 cells assessed as T-cell factor level after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50498898(CHEMBL3736494)
Affinity DataIC50: 60nMAssay Description:Inhibition of TNKS2 (unknown origin) by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50498905(CHEMBL3736012)
Affinity DataIC50: 60nMAssay Description:Inhibition of TNKS2 (unknown origin) by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50498900(CHEMBL3736145)
Affinity DataIC50: 60nMAssay Description:Inhibition of TNKS2 (unknown origin) by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50498903(CHEMBL3735964)
Affinity DataIC50: 60nMAssay Description:Inhibition of TNKS2 (unknown origin) by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50498904(CHEMBL3734991)
Affinity DataIC50: 60nMAssay Description:Inhibition of TNKS2 (unknown origin) by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50498901(CHEMBL3735517)
Affinity DataIC50: 60nMAssay Description:Inhibition of TNKS2 (unknown origin) by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50498897(CHEMBL3734971)
Affinity DataIC50: 60nMAssay Description:Inhibition of TNKS2 (unknown origin) by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50498899(CHEMBL3736005)
Affinity DataIC50: 93nMAssay Description:Inhibition of TNKS2 (unknown origin) by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1/tankyrase-2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50498901(CHEMBL3735517)
Affinity DataEC50:  127nMAssay Description:Inhibition of Tankyrase in human DLD1 cells assessed as T-cell factor level after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50321122(2-Ethylquinazolin-4(3H)-one | CHEMBL1163173)
Affinity DataIC50: 140nMAssay Description:Inhibition of TNKS1 (unknown origin) by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50321122(2-Ethylquinazolin-4(3H)-one | CHEMBL1163173)
Affinity DataIC50: 200nMAssay Description:Inhibition of TNKS2 (unknown origin) by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1/tankyrase-2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50498898(CHEMBL3736494)
Affinity DataEC50:  320nMAssay Description:Inhibition of Tankyrase in human DLD1 cells assessed as T-cell factor level after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1/tankyrase-2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50498897(CHEMBL3734971)
Affinity DataEC50:  341nMAssay Description:Inhibition of Tankyrase in human DLD1 cells assessed as T-cell factor level after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1/tankyrase-2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50498899(CHEMBL3736005)
Affinity DataEC50:  810nMAssay Description:Inhibition of Tankyrase in human DLD1 cells assessed as T-cell factor level after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50498902(CHEMBL1527375)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of TNKS1 (unknown origin) by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50498902(CHEMBL1527375)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of TNKS2 (unknown origin) by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed