Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50022527
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM257207(US9493440, 51)
Affinity DataIC50: 0.760nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM257207(US9493440, 51)
Affinity DataIC50: 1.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetDual specificity protein kinase CLK4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM257207(US9493440, 51)
Affinity DataIC50: 225nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 14(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM257207(US9493440, 51)
Affinity DataIC50: 244nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM257207(US9493440, 51)
Affinity DataIC50: 428nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetDual specificity protein kinase CLK2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM257207(US9493440, 51)
Affinity DataIC50: 605nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetDual specificity protein kinase TTK(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM257207(US9493440, 51)
Affinity DataIC50: 935nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM257207(US9493440, 51)
Affinity DataIC50: 1.20E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM257207(US9493440, 51)
Affinity DataIC50: 3.80E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM257207(US9493440, 51)
Affinity DataIC50: 6.40E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM257207(US9493440, 51)
Affinity DataIC50: 6.50E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM257207(US9493440, 51)
Affinity DataKi:  3.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed