Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50046784
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | S-[1-(adenin-9-yl)-1,5-dideoxy-beta-D-rib...)
Affinity DataIC50: 500nMAssay Description:Inhibition of PRMT1 (unknown origin) using biotinylated histone H4-derived peptide as substrate after 60 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50130929(CHEMBL3633189)
Affinity DataKi:  1.70E+3nMAssay Description:Non-competitive inhibition of PRMT1 (unknown origin) using biotinylated histone H4-derived peptide as substrate by Michaelis-Menten kinetic equation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50130929(CHEMBL3633189)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of PRMT1 (unknown origin) using biotinylated histone H4-derived peptide as substrate after 60 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50130932(CHEMBL3633187)
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of PRMT1 (unknown origin) using biotinylated histone H4-derived peptide as substrate after 60 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50130929(CHEMBL3633189)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PRMT4 (unknown origin) using biotinylated histone H4-derived peptide as substrate after 60 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50130931(CHEMBL3633188)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of PRMT1 (unknown origin) using biotinylated histone H4-derived peptide as substrate after 60 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50446401(CHEMBL3109656)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of PRMT1 (unknown origin) using biotinylated histone H4-derived peptide as substrate after 60 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50130930(CHEMBL3633190)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of PRMT1 (unknown origin) using biotinylated histone H4-derived peptide as substrate after 60 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50130933(CHEMBL3633186)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of PRMT1 (unknown origin) using biotinylated histone H4-derived peptide as substrate after 60 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50130929(CHEMBL3633189)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PRMT6 (unknown origin) using biotinylated histone H4-derived peptide as substrate after 60 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50130929(CHEMBL3633189)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PRMT5 (unknown origin) using biotinylated histone H4-derived peptide as substrate after 60 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed