Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50006339
LigandPNGBDBM50250018(PACAP27 | CHEMBL524852)
Affinity DataIC50: 4.60nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human PAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVasoactive intestinal polypeptide receptor 1(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50250018(PACAP27 | CHEMBL524852)
Affinity DataIC50: 5.90nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVasoactive intestinal polypeptide receptor 1(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50498951(CHEMBL3736134)
Affinity DataIC50: 9nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVasoactive intestinal polypeptide receptor 1(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50498951(CHEMBL3736134)
Affinity DataIC50: 9.30nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVasoactive intestinal polypeptide receptor 2(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50250018(PACAP27 | CHEMBL524852)
Affinity DataIC50: 10nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC2 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVasoactive intestinal polypeptide receptor 1(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50498950(CHEMBL3736230)
Affinity DataIC50: 11nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVasoactive intestinal polypeptide receptor 1(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50498950(CHEMBL3736230)
Affinity DataIC50: 12nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVasoactive intestinal polypeptide receptor 1(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50250074([Bip6]PACAP27 | CHEMBL507480)
Affinity DataIC50: 14nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVasoactive intestinal polypeptide receptor 2(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50250074([Bip6]PACAP27 | CHEMBL507480)
Affinity DataIC50: 23nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC2 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVasoactive intestinal polypeptide receptor 2(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50498951(CHEMBL3736134)
Affinity DataIC50: 36nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC2 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVasoactive intestinal polypeptide receptor 2(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50498951(CHEMBL3736134)
Affinity DataIC50: 36nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC2 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
LigandPNGBDBM50498950(CHEMBL3736230)
Affinity DataIC50: 44.7nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human PAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
LigandPNGBDBM50498950(CHEMBL3736230)
Affinity DataIC50: 45nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human PAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVasoactive intestinal polypeptide receptor 2(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50498950(CHEMBL3736230)
Affinity DataIC50: 53nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC2 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVasoactive intestinal polypeptide receptor 2(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50498950(CHEMBL3736230)
Affinity DataIC50: 54nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC2 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
LigandPNGBDBM50498951(CHEMBL3736134)
Affinity DataIC50: 57nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human PAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
LigandPNGBDBM50498951(CHEMBL3736134)
Affinity DataIC50: 58nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human PAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed