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Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50046810
TargetHistone deacetylase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132484(CHEMBL3633769)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of human HDAC in HeLa cell nuclear extract by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132484(CHEMBL3633769)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human recombinant HDAC1 by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132403(CHEMBL3633765)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of human HDAC in HeLa cell nuclear extract by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132484(CHEMBL3633769)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of human recombinant HDAC8 by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132345(CHEMBL3633761)
Affinity DataIC50: 5.40nMAssay Description:Inhibition of human HDAC in HeLa cell nuclear extract by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132484(CHEMBL3633769)
Affinity DataIC50: 6.80nMAssay Description:Inhibition of human recombinant HDAC2 by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132488(CHEMBL3633773)
Affinity DataIC50: 8.40nMAssay Description:Inhibition of human HDAC in HeLa cell nuclear extract by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human HDAC in HeLa cell nuclear extract by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132482(CHEMBL3633768)
Affinity DataIC50: 14nMAssay Description:Inhibition of human HDAC in HeLa cell nuclear extract by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132389(CHEMBL3633764)
Affinity DataIC50: 15nMAssay Description:Inhibition of human HDAC in HeLa cell nuclear extract by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132344(CHEMBL3633760)
Affinity DataIC50: 17nMAssay Description:Inhibition of human HDAC in HeLa cell nuclear extract by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132487(CHEMBL3633772)
Affinity DataIC50: 21nMAssay Description:Inhibition of human HDAC in HeLa cell nuclear extract by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132484(CHEMBL3633769)
Affinity DataIC50: 26nMAssay Description:Inhibition of human recombinant HDAC6 by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132486(CHEMBL3633771)
Affinity DataIC50: 57nMAssay Description:Inhibition of human HDAC in HeLa cell nuclear extract by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM21(VANDETANIB | N-(4-bromo-2-fluorophenyl)-6-methoxy-...)
Affinity DataIC50: 62nMAssay Description:Inhibition VEGFR2 (unknown origin) for 30 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132484(CHEMBL3633769)
Affinity DataIC50: 84nMAssay Description:Inhibition VEGFR2 (unknown origin) for 30 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132480(CHEMBL3633767)
Affinity DataIC50: 86nMAssay Description:Inhibition of human HDAC in HeLa cell nuclear extract by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132347(CHEMBL3633763)
Affinity DataIC50: 97nMAssay Description:Inhibition of human HDAC in HeLa cell nuclear extract by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132482(CHEMBL3633768)
Affinity DataIC50: 115nMAssay Description:Inhibition VEGFR2 (unknown origin) for 30 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132343(CHEMBL3633759)
Affinity DataIC50: 121nMAssay Description:Inhibition of human HDAC in HeLa cell nuclear extract by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132480(CHEMBL3633767)
Affinity DataIC50: 138nMAssay Description:Inhibition VEGFR2 (unknown origin) for 30 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132479(CHEMBL3633766)
Affinity DataIC50: 215nMAssay Description:Inhibition of human HDAC in HeLa cell nuclear extract by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132485(CHEMBL3633770)
Affinity DataIC50: 348nMAssay Description:Inhibition of human HDAC in HeLa cell nuclear extract by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132343(CHEMBL3633759)
Affinity DataIC50: 352nMAssay Description:Inhibition VEGFR2 (unknown origin) for 30 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132479(CHEMBL3633766)
Affinity DataIC50: 370nMAssay Description:Inhibition VEGFR2 (unknown origin) for 30 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132389(CHEMBL3633764)
Affinity DataIC50: 415nMAssay Description:Inhibition VEGFR2 (unknown origin) for 30 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132347(CHEMBL3633763)
Affinity DataIC50: 434nMAssay Description:Inhibition VEGFR2 (unknown origin) for 30 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132403(CHEMBL3633765)
Affinity DataIC50: 462nMAssay Description:Inhibition VEGFR2 (unknown origin) for 30 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132342(CHEMBL3633758)
Affinity DataIC50: 476nMAssay Description:Inhibition VEGFR2 (unknown origin) for 30 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132345(CHEMBL3633761)
Affinity DataIC50: 501nMAssay Description:Inhibition VEGFR2 (unknown origin) for 30 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132346(CHEMBL3633762)
Affinity DataIC50: 531nMAssay Description:Inhibition of human HDAC in HeLa cell nuclear extract by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132344(CHEMBL3633760)
Affinity DataIC50: 613nMAssay Description:Inhibition VEGFR2 (unknown origin) for 30 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132346(CHEMBL3633762)
Affinity DataIC50: 625nMAssay Description:Inhibition VEGFR2 (unknown origin) for 30 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132342(CHEMBL3633758)
Affinity DataIC50: 645nMAssay Description:Inhibition of human HDAC in HeLa cell nuclear extract by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132485(CHEMBL3633770)
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition VEGFR2 (unknown origin) for 30 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132486(CHEMBL3633771)
Affinity DataIC50: 2.14E+3nMAssay Description:Inhibition VEGFR2 (unknown origin) for 30 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132488(CHEMBL3633773)
Affinity DataIC50: 2.45E+3nMAssay Description:Inhibition VEGFR2 (unknown origin) for 30 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50132487(CHEMBL3633772)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition VEGFR2 (unknown origin) for 30 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition VEGFR2 (unknown origin) for 30 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM21(VANDETANIB | N-(4-bromo-2-fluorophenyl)-6-methoxy-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human HDAC in HeLa cell nuclear extract by fluorometric assay using Fluor de Lys substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2016
Entry Details Article
PubMed