Report error Found 79 Enz. Inhib. hit(s) with all data for entry = 50006356
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
University of Tours
Curated by ChEMBL
University of Tours
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of full length human GST-tagged RIPK3 expressed in Spodoptera frugiperda Sf9 cells after 30 mins by scintillation and luminescence countin...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
University of Tours
Curated by ChEMBL
University of Tours
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of full length human GST-tagged RIPK3 expressed in Spodoptera frugiperda Sf9 cells after 30 mins by scintillation and luminescence countin...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
University of Tours
Curated by ChEMBL
University of Tours
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:Inhibition of full length human GST-tagged RIPK3 expressed in Spodoptera frugiperda Sf9 cells after 30 mins by scintillation and luminescence countin...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
University of Tours
Curated by ChEMBL
University of Tours
Curated by ChEMBL
Affinity DataIC50: 880nMAssay Description:Inhibition of full length human GST-tagged RIPK3 expressed in Spodoptera frugiperda Sf9 cells after 30 mins by scintillation and luminescence countin...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
University of Tours
Curated by ChEMBL
University of Tours
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of full length human GST-tagged RIPK3 expressed in Spodoptera frugiperda Sf9 cells after 30 mins by scintillation and luminescence countin...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
University of Tours
Curated by ChEMBL
University of Tours
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of full length human GST-tagged RIPK3 expressed in Spodoptera frugiperda Sf9 cells after 30 mins by scintillation and luminescence countin...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of porcine brain GSK-3 alpha/beta using GS-1 substrate after 30 mins by scintillation and luminescence counting method in the presence of ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
University of Tours
Curated by ChEMBL
University of Tours
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of full length human GST-tagged RIPK3 expressed in Spodoptera frugiperda Sf9 cells after 30 mins by scintillation and luminescence countin...More data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of porcine brain GSK-3 alpha/beta using GS-1 substrate after 30 mins by scintillation and luminescence counting method in the presence of ...More data for this Ligand-Target Pair
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of human recombinant haspin kinase domain expressed in Escherichia coli BL21-KRX using histone H3 (1 to 21) peptide substrate after 30 min...More data for this Ligand-Target Pair
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of porcine brain GSK-3 alpha/beta using GS-1 substrate after 30 mins by scintillation and luminescence counting method in the presence of ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
University of Tours
Curated by ChEMBL
University of Tours
Curated by ChEMBL
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of full length human GST-tagged RIPK3 expressed in Spodoptera frugiperda Sf9 cells after 30 mins by scintillation and luminescence countin...More data for this Ligand-Target Pair
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of porcine brain GSK-3 alpha/beta using GS-1 substrate after 30 mins by scintillation and luminescence counting method in the presence of ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
University of Tours
Curated by ChEMBL
University of Tours
Curated by ChEMBL
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of full length human GST-tagged RIPK3 expressed in Spodoptera frugiperda Sf9 cells after 30 mins by scintillation and luminescence countin...More data for this Ligand-Target Pair
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of porcine brain GSK-3 alpha/beta using GS-1 substrate after 30 mins by scintillation and luminescence counting method in the presence of ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of porcine brain GSK-3 alpha/beta using GS-1 substrate after 30 mins by scintillation and luminescence counting method in the presence of ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
University of Tours
Curated by ChEMBL
University of Tours
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of full length human GST-tagged RIPK3 expressed in Spodoptera frugiperda Sf9 cells after 30 mins by scintillation and luminescence countin...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant haspin kinase domain expressed in Escherichia coli BL21-KRX using histone H3 (1 to 21) peptide substrate after 30 min...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
University of Tours
Curated by ChEMBL
University of Tours
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of full length human GST-tagged RIPK3 expressed in Spodoptera frugiperda Sf9 cells after 30 mins by scintillation and luminescence countin...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 expressed in Escherichia coli using histone H1 substrate after 30 mins by scintillation and luminescence cou...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
University of Tours
Curated by ChEMBL
University of Tours
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of full length human GST-tagged RIPK3 expressed in Spodoptera frugiperda Sf9 cells after 30 mins by scintillation and luminescence countin...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
University of Tours
Curated by ChEMBL
University of Tours
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of full length human GST-tagged RIPK3 expressed in Spodoptera frugiperda Sf9 cells after 30 mins by scintillation and luminescence countin...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 expressed in Escherichia coli using histone H1 substrate after 30 mins by scintillation and luminescence cou...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 expressed in Escherichia coli using histone H1 substrate after 30 mins by scintillation and luminescence cou...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 expressed in Escherichia coli using histone H1 substrate after 30 mins by scintillation and luminescence cou...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of porcine brain GSK-3 alpha/beta using GS-1 substrate after 30 mins by scintillation and luminescence counting method in the presence of ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of porcine brain GSK-3 alpha/beta using GS-1 substrate after 30 mins by scintillation and luminescence counting method in the presence of ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant haspin kinase domain expressed in Escherichia coli BL21-KRX using histone H3 (1 to 21) peptide substrate after 30 min...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant haspin kinase domain expressed in Escherichia coli BL21-KRX using histone H3 (1 to 21) peptide substrate after 30 min...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 expressed in Escherichia coli using histone H1 substrate after 30 mins by scintillation and luminescence cou...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of porcine brain GSK-3 alpha/beta using GS-1 substrate after 30 mins by scintillation and luminescence counting method in the presence of ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of porcine brain GSK-3 alpha/beta using GS-1 substrate after 30 mins by scintillation and luminescence counting method in the presence of ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
University of Tours
Curated by ChEMBL
University of Tours
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of full length human GST-tagged RIPK3 expressed in Spodoptera frugiperda Sf9 cells after 30 mins by scintillation and luminescence countin...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant haspin kinase domain expressed in Escherichia coli BL21-KRX using histone H3 (1 to 21) peptide substrate after 30 min...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant haspin kinase domain expressed in Escherichia coli BL21-KRX using histone H3 (1 to 21) peptide substrate after 30 min...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 expressed in Escherichia coli using histone H1 substrate after 30 mins by scintillation and luminescence cou...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
University of Tours
Curated by ChEMBL
University of Tours
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of full length human GST-tagged RIPK3 expressed in Spodoptera frugiperda Sf9 cells after 30 mins by scintillation and luminescence countin...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant haspin kinase domain expressed in Escherichia coli BL21-KRX using histone H3 (1 to 21) peptide substrate after 30 min...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant haspin kinase domain expressed in Escherichia coli BL21-KRX using histone H3 (1 to 21) peptide substrate after 30 min...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of porcine brain GSK-3 alpha/beta using GS-1 substrate after 30 mins by scintillation and luminescence counting method in the presence of ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 expressed in Escherichia coli using histone H1 substrate after 30 mins by scintillation and luminescence cou...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 expressed in Escherichia coli using histone H1 substrate after 30 mins by scintillation and luminescence cou...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant haspin kinase domain expressed in Escherichia coli BL21-KRX using histone H3 (1 to 21) peptide substrate after 30 min...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 expressed in Escherichia coli using histone H1 substrate after 30 mins by scintillation and luminescence cou...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 expressed in Escherichia coli using histone H1 substrate after 30 mins by scintillation and luminescence cou...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 expressed in Escherichia coli using histone H1 substrate after 30 mins by scintillation and luminescence cou...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 expressed in Escherichia coli using histone H1 substrate after 30 mins by scintillation and luminescence cou...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 expressed in Escherichia coli using histone H1 substrate after 30 mins by scintillation and luminescence cou...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 expressed in Escherichia coli using histone H1 substrate after 30 mins by scintillation and luminescence cou...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 expressed in Escherichia coli using histone H1 substrate after 30 mins by scintillation and luminescence cou...More data for this Ligand-Target Pair
