Report error Found 59 Enz. Inhib. hit(s) with all data for entry = 50046833
Affinity DataIC50: 4.16E+3nMAssay Description:Antagonist activity at human muscarinic M3 receptor expressed in HEK293 cells assessed as inhibition of carbachol-induced inositol monophosphate accu...More data for this Ligand-Target Pair
Affinity DataIC50: 4.17E+3nMAssay Description:Antagonist activity at human muscarinic M3 receptor expressed in HEK293 cells assessed as inhibition of carbachol-induced inositol monophosphate accu...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 5.50E+3nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 5.50E+3nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 6.17E+3nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 6.17E+3nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 9.33E+3nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 9.33E+3nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 2.13E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 2.14E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 2.19E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 2.19E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
Affinity DataIC50: 2.75E+4nMAssay Description:Antagonist activity at human muscarinic M3 receptor expressed in HEK293 cells assessed as inhibition of carbachol-induced inositol monophosphate accu...More data for this Ligand-Target Pair
Affinity DataIC50: 2.75E+4nMAssay Description:Antagonist activity at human muscarinic M3 receptor expressed in HEK293 cells assessed as inhibition of carbachol-induced inositol monophosphate accu...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 3.98E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 3.98E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
Affinity DataIC50: 4.17E+4nMAssay Description:Antagonist activity at rat mGluR5 expressed in CHO cells assessed as inhibition of L-glutamate-induced inositol monophosphate accumulation after 1 hr...More data for this Ligand-Target Pair
Affinity DataIC50: 4.17E+4nMAssay Description:Antagonist activity at rat mGluR5 expressed in CHO cells assessed as inhibition of L-glutamate-induced inositol monophosphate accumulation after 1 hr...More data for this Ligand-Target Pair
Affinity DataIC50: 5.12E+4nMAssay Description:Antagonist activity at human muscarinic M3 receptor expressed in HEK293 cells assessed as inhibition of carbachol-induced inositol monophosphate accu...More data for this Ligand-Target Pair
Affinity DataIC50: 5.13E+4nMAssay Description:Antagonist activity at human muscarinic M3 receptor expressed in HEK293 cells assessed as inhibition of carbachol-induced inositol monophosphate accu...More data for this Ligand-Target Pair
Affinity DataIC50: 5.13E+4nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced inositol monophosphate accumulation...More data for this Ligand-Target Pair
Affinity DataIC50: 5.13E+4nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced inositol monophosphate accumulation...More data for this Ligand-Target Pair
Affinity DataIC50: 5.62E+4nMAssay Description:Antagonist activity at rat CaSR expressed in HEK293 cells assessed as inhibition of Ca2+-induced inositol monophosphate accumulation after 1 hr by FR...More data for this Ligand-Target Pair
Affinity DataIC50: 5.62E+4nMAssay Description:Antagonist activity at rat CaSR expressed in HEK293 cells assessed as inhibition of Ca2+-induced inositol monophosphate accumulation after 1 hr by FR...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 5.73E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
Affinity DataIC50: 5.75E+4nMAssay Description:Antagonist activity at human muscarinic M3 receptor expressed in HEK293 cells assessed as inhibition of carbachol-induced inositol monophosphate accu...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 5.75E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
Affinity DataIC50: 5.75E+4nMAssay Description:Antagonist activity at human muscarinic M3 receptor expressed in HEK293 cells assessed as inhibition of carbachol-induced inositol monophosphate accu...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 6.61E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 6.61E+4nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 1.32E+5nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 1.32E+5nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
Affinity DataIC50: 2.09E+5nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced inositol monophosphate accumulation...More data for this Ligand-Target Pair
Affinity DataIC50: 2.09E+5nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced inositol monophosphate accumulation...More data for this Ligand-Target Pair
Affinity DataIC50: 2.14E+5nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced inositol monophosphate accumulation...More data for this Ligand-Target Pair
Affinity DataIC50: 2.14E+5nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced inositol monophosphate accumulation...More data for this Ligand-Target Pair
Affinity DataIC50: 2.24E+5nMAssay Description:Antagonist activity at rat mGluR5 expressed in CHO cells assessed as inhibition of L-glutamate-induced inositol monophosphate accumulation after 1 hr...More data for this Ligand-Target Pair
Affinity DataIC50: 2.24E+5nMAssay Description:Antagonist activity at rat mGluR5 expressed in CHO cells assessed as inhibition of L-glutamate-induced inositol monophosphate accumulation after 1 hr...More data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+5nMAssay Description:Antagonist activity at rat CaSR expressed in HEK293 cells assessed as inhibition of Ca2+-induced inositol monophosphate accumulation after 1 hr by FR...More data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+5nMAssay Description:Antagonist activity at rat CaSR expressed in HEK293 cells assessed as inhibition of Ca2+-induced inositol monophosphate accumulation after 1 hr by FR...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 2.45E+5nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 2.48E+5nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 2.56E+5nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
TargetG-protein coupled receptor family C group 6 member A(Mouse)
University of Copenhagen
Curated by ChEMBL
University of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 2.57E+5nMAssay Description:Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat...More data for this Ligand-Target Pair
Affinity DataIC50: 2.63E+5nMAssay Description:Antagonist activity at rat mGluR5 expressed in CHO cells assessed as inhibition of L-glutamate-induced inositol monophosphate accumulation after 1 hr...More data for this Ligand-Target Pair
Affinity DataIC50: 2.63E+5nMAssay Description:Antagonist activity at rat mGluR5 expressed in CHO cells assessed as inhibition of L-glutamate-induced inositol monophosphate accumulation after 1 hr...More data for this Ligand-Target Pair
Affinity DataIC50: 2.69E+5nMAssay Description:Antagonist activity at rat mGluR5 expressed in CHO cells assessed as inhibition of L-glutamate-induced inositol monophosphate accumulation after 1 hr...More data for this Ligand-Target Pair
Affinity DataIC50: 2.69E+5nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced inositol monophosphate accumulation...More data for this Ligand-Target Pair
Affinity DataIC50: 2.69E+5nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced inositol monophosphate accumulation...More data for this Ligand-Target Pair
Affinity DataIC50: 2.69E+5nMAssay Description:Antagonist activity at rat mGluR5 expressed in CHO cells assessed as inhibition of L-glutamate-induced inositol monophosphate accumulation after 1 hr...More data for this Ligand-Target Pair
