Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50046761
TargetLIM domain kinase 1(Human)
Shanghai Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50130039(CHEMBL3629276)
Affinity DataIC50: 10nMAssay Description:Inhibition of LIMK1 (unknown origin) using 1 uM cofilin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetLIM domain kinase 1(Human)
Shanghai Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50130038(CHEMBL3629277)
Affinity DataIC50: 11nMAssay Description:Inhibition of LIMK1 (unknown origin) using 1 uM cofilin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetLIM domain kinase 1(Human)
Shanghai Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50130037(CHEMBL3629278)
Affinity DataIC50: 19nMAssay Description:Inhibition of LIMK1 (unknown origin) using 1 uM cofilin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetLIM domain kinase 1(Human)
Shanghai Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50130036(CHEMBL3629279)
Affinity DataIC50: 55nMAssay Description:Inhibition of LIMK1 (unknown origin) using 1 uM cofilin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetLIM domain kinase 1(Human)
Shanghai Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50130035(CHEMBL3629280)
Affinity DataIC50: 85nMAssay Description:Inhibition of LIMK1 (unknown origin) using 1 uM cofilin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Shanghai Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50130036(CHEMBL3629279)
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of ROCK2 (unknown origin) after 4 hrs using 1 uM STK2 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Shanghai Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50130037(CHEMBL3629278)
Affinity DataIC50: 2.01E+3nMAssay Description:Inhibition of ROCK2 (unknown origin) after 4 hrs using 1 uM STK2 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Shanghai Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50130038(CHEMBL3629277)
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of ROCK2 (unknown origin) after 4 hrs using 1 uM STK2 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Shanghai Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50130035(CHEMBL3629280)
Affinity DataIC50: 4.51E+3nMAssay Description:Inhibition of ROCK2 (unknown origin) after 4 hrs using 1 uM STK2 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Shanghai Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50130039(CHEMBL3629276)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of ROCK2 (unknown origin) after 4 hrs using 1 uM STK2 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed