Compile Data Set for Download or QSAR
Report error Found 82 Enz. Inhib. hit(s) with all data for entry = 50006495
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500324(CHEMBL3747448)
Affinity DataIC50: 6nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500325(Cb 5083 | Cb-5083)
Affinity DataIC50: 11nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500319(CHEMBL3746179)
Affinity DataIC50: 15nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500347(CHEMBL3747049)
Affinity DataIC50: 23nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500310(CHEMBL3747647)
Affinity DataIC50: 40nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163143(US9062026, Table III, Compound 71)
Affinity DataIC50: 43nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163134(US9062026, Table III, Compound 62)
Affinity DataIC50: 47nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163144(US9062026, Table III, Compound 72)
Affinity DataIC50: 68nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500321(CHEMBL3745888)
Affinity DataIC50: 71nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500323(CHEMBL3746353)
Affinity DataIC50: 76nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500318(CHEMBL3746650)
Affinity DataIC50: 95nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500339(CHEMBL3747498)
Affinity DataIC50: 98nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500316(CHEMBL3746000)
Affinity DataIC50: 144nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163082(US9062026, Table III, Compound 10)
Affinity DataIC50: 145nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500337(CHEMBL3747075)
Affinity DataIC50: 149nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163080(US9062026, Table III, Compound 8)
Affinity DataIC50: 152nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163136(US9062026, Table III, Compound 79 | US9062026, Tab...)
Affinity DataIC50: 153nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163092(US9062026, Table III, Compound 20)
Affinity DataIC50: 180nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163115(US9062026, Table III, Compound 43)
Affinity DataIC50: 192nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500320(CHEMBL3747639)
Affinity DataIC50: 215nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163098(US9062026, Table III, Compound 26)
Affinity DataIC50: 227nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163097(US9062026, Table III, Compound 25)
Affinity DataIC50: 233nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500312(CHEMBL3746787)
Affinity DataIC50: 248nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500324(CHEMBL3747448)
Affinity DataIC50: 250nMAssay Description:Inhibition of p97 ATPase in human A549 cells assessed as reduction in p62 protein incubated for 6 hrs by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500335(CHEMBL3746988)
Affinity DataIC50: 304nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500309(CHEMBL3745805)
Affinity DataIC50: 342nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500307(CHEMBL3746833)
Affinity DataIC50: 367nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500331(CHEMBL3220939)
Affinity DataIC50: 370nMAssay Description:Inhibition of p97 ATPase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163139(US9062026, Table III, Compound 67)
Affinity DataIC50: 370nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500327(CHEMBL3746037)
Affinity DataIC50: 425nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163135(US9062026, Table III, Compound 63)
Affinity DataIC50: 445nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500325(Cb 5083 | Cb-5083)
Affinity DataIC50: 490nMAssay Description:Inhibition of p97 ATPase in human A549 cells assessed as reduction in p62 protein incubated for 6 hrs by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500325(Cb 5083 | Cb-5083)
Affinity DataIC50: 500nMAssay Description:Inhibition of DNAPK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500324(CHEMBL3747448)
Affinity DataIC50: 500nMAssay Description:Inhibition of p97 ATPase in human A549 cells assessed as accumulation of K48 poly-ubiquitinated proteins incubated for 6 hrs by immunofluorescence as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500324(CHEMBL3747448)
Affinity DataIC50: 580nMAssay Description:Inhibition of p97 ATPase in human A549 cells assessed as accumulation of CHOP poly-ubiquitinated proteins incubated for 6 hrs by immunofluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500332(CHEMBL3747140)
Affinity DataIC50: 632nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500315(CHEMBL3747371)
Affinity DataIC50: 648nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500306(CHEMBL3747138)
Affinity DataIC50: 651nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500325(Cb 5083 | Cb-5083)
Affinity DataIC50: 680nMAssay Description:Inhibition of p97 ATPase in human A549 cells assessed as accumulation of K48 poly-ubiquitinated proteins incubated for 6 hrs by immunofluorescence as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163145(US9062026, Table III, Compound 73)
Affinity DataIC50: 795nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500322(CHEMBL3746912)
Affinity DataIC50: 815nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163086(US9062026, Table III, Compound 14)
Affinity DataIC50: 907nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500325(Cb 5083 | Cb-5083)
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of p97 ATPase in human A549 cells assessed as accumulation of CHOP poly-ubiquitinated proteins incubated for 6 hrs by immunofluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163106(US9062026, Table III, Compound 34)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500310(CHEMBL3747647)
Affinity DataIC50: 1.79E+3nMAssay Description:Inhibition of p97 ATPase in human A549 cells assessed as accumulation of K48 poly-ubiquitinated proteins incubated for 6 hrs by immunofluorescence as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500310(CHEMBL3747647)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of p97 ATPase in human A549 cells assessed as reduction in p62 protein incubated for 6 hrs by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500338(CHEMBL3747194)
Affinity DataIC50: 2.08E+3nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500310(CHEMBL3747647)
Affinity DataIC50: 2.86E+3nMAssay Description:Inhibition of p97 ATPase in human A549 cells assessed as accumulation of CHOP poly-ubiquitinated proteins incubated for 6 hrs by immunofluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM50500305(CHEMBL3747511)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
Cleave Biosciences

Curated by ChEMBL
LigandPNGBDBM163114(US9062026, Table III, Compound 42)
Affinity DataIC50: 3.13E+3nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
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