Compile Data Set for Download or QSAR
Report error Found 136 Enz. Inhib. hit(s) with all data for entry = 50046907
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50426075(CHEMBL473104)
Affinity DataIC50: 180nMAssay Description:Inhibition of mouse GAT1 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 3(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50039246((S)-1-(2-(tris(4-methoxyphenyl)methoxy)ethyl)piper...)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of mouse GAT3 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM90787(SMR000326834 | cid_11957555 | GUVACINE | MLS000859...)
Affinity DataIC50: 2.09E+4nMAssay Description:Inhibition of mouse GAT1 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50039246((S)-1-(2-(tris(4-methoxyphenyl)methoxy)ethyl)piper...)
Affinity DataIC50: 2.19E+4nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM90787(SMR000326834 | cid_11957555 | GUVACINE | MLS000859...)
Affinity DataIC50: 7.24E+4nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent betaine transporter(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137093(CHEMBL3754254)
Affinity DataIC50: 1.03E+5nMAssay Description:Inhibition of mouse BGT1 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent betaine transporter(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50136963(CHEMBL3753393)
Affinity DataIC50: 1.03E+5nMAssay Description:Inhibition of mouse BGT1 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 3(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM90787(SMR000326834 | cid_11957555 | GUVACINE | MLS000859...)
Affinity DataIC50: 1.15E+5nMAssay Description:Inhibition of mouse GAT3 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent betaine transporter(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50136988(CHEMBL3753440)
Affinity DataIC50: 1.64E+5nMAssay Description:Inhibition of mouse BGT1 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50039246((S)-1-(2-(tris(4-methoxyphenyl)methoxy)ethyl)piper...)
Affinity DataIC50: 1.99E+5nMAssay Description:Inhibition of mouse GAT1 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137073(CHEMBL3753682)
Affinity DataIC50: 2.33E+5nMAssay Description:Inhibition of mouse GAT1 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50136963(CHEMBL3753393)
Affinity DataIC50: 3.71E+5nMAssay Description:Inhibition of mouse GAT1 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137093(CHEMBL3754254)
Affinity DataIC50: 3.71E+5nMAssay Description:Inhibition of mouse GAT1 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 3(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137074(CHEMBL3752644)
Affinity DataIC50: 6.75E+5nMAssay Description:Inhibition of mouse GAT3 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 3(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50136988(CHEMBL3753440)
Affinity DataIC50: 9.33E+5nMAssay Description:Inhibition of mouse GAT3 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50136881(CHEMBL3752875)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50136904(CHEMBL3752268)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50136963(CHEMBL3753393)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50136968(CHEMBL3753545)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50136970(CHEMBL3753634)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50136977(CHEMBL3753899)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50136982(CHEMBL3752003)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50136988(CHEMBL3753440)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137023(CHEMBL3753364)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137025(CHEMBL3754424)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137071(CHEMBL3751979)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137072(CHEMBL3752695)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137073(CHEMBL3753682)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137074(CHEMBL3752644)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137075(CHEMBL3753896)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137076(CHEMBL3754490)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137077(CHEMBL3754503)
Affinity DataIC50: 2.33E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137080(CHEMBL3753151)
Affinity DataIC50: 3.23E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137081(CHEMBL3753338)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137082(CHEMBL3752449)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137083(CHEMBL3752733)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137084(CHEMBL3753616)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137085(CHEMBL3752032)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137086(CHEMBL3752080)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137087(CHEMBL3752039)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50426075(CHEMBL473104)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 3(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137088(CHEMBL1887095)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition of mouse GAT3 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 3(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137089(CHEMBL3753828)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition of mouse GAT3 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 3(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137090(CHEMBL3754441)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT3 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 3(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137091(CHEMBL3752545)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT3 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 3(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137092(CHEMBL3753554)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition of mouse GAT3 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 3(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50137093(CHEMBL3754254)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT3 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 3(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50136881(CHEMBL3752875)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT3 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 3(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50136904(CHEMBL3752268)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT3 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 3(Mouse)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50136963(CHEMBL3753393)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT3 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
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