Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50046893
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135269(CHEMBL3745775)
Affinity DataKi:  0.830nMAssay Description:Inhibition of human recombinant hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135268(CHEMBL3747482)
Affinity DataKi:  1nMAssay Description:Inhibition of human recombinant hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50032936(CHEMBL3356589)
Affinity DataKi:  1.5nMAssay Description:Inhibition of human recombinant hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135270(CHEMBL3747468)
Affinity DataKi:  2.90nMAssay Description:Inhibition of human recombinant hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135275(CHEMBL3746517)
Affinity DataKi:  2.90nMAssay Description:Inhibition of human recombinant hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135274(CHEMBL404190)
Affinity DataKi:  3.40nMAssay Description:Inhibition of human recombinant hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein homolog(Mouse)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135269(CHEMBL3745775)
Affinity DataKi:  8nMAssay Description:Inhibition of mouse recombinant matriptase using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein homolog(Mouse)
Korea University

Curated by ChEMBL
LigandPNGBDBM50032936(CHEMBL3356589)
Affinity DataKi:  10nMAssay Description:Inhibition of mouse recombinant matriptase using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein homolog(Mouse)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135268(CHEMBL3747482)
Affinity DataKi:  11nMAssay Description:Inhibition of mouse recombinant matriptase using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein homolog(Mouse)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135270(CHEMBL3747468)
Affinity DataKi:  11nMAssay Description:Inhibition of mouse recombinant matriptase using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135272(CHEMBL3747618)
Affinity DataKi:  22nMAssay Description:Inhibition of human recombinant hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135271(CHEMBL3747575)
Affinity DataKi:  22nMAssay Description:Inhibition of human recombinant hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein homolog(Mouse)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135275(CHEMBL3746517)
Affinity DataKi:  177nMAssay Description:Inhibition of mouse recombinant matriptase using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein homolog(Mouse)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135274(CHEMBL404190)
Affinity DataKi:  227nMAssay Description:Inhibition of mouse recombinant matriptase using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein homolog(Mouse)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135272(CHEMBL3747618)
Affinity DataKi:  246nMAssay Description:Inhibition of mouse recombinant matriptase using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein homolog(Mouse)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135271(CHEMBL3747575)
Affinity DataKi:  334nMAssay Description:Inhibition of mouse recombinant matriptase using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135273(CHEMBL3747752)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human recombinant hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135276(CHEMBL3746062)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human recombinant hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135277(CHEMBL3746635)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human recombinant hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135278(CHEMBL3747693)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human recombinant hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein homolog(Mouse)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135273(CHEMBL3747752)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of mouse recombinant matriptase using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein homolog(Mouse)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135276(CHEMBL3746062)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of mouse recombinant matriptase using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein homolog(Mouse)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135277(CHEMBL3746635)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of mouse recombinant matriptase using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein homolog(Mouse)
Korea University

Curated by ChEMBL
LigandPNGBDBM50135278(CHEMBL3747693)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of mouse recombinant matriptase using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 15 to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed