Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50047115
LigandPNGBDBM25045(CHEMBL538346 | mTOR Inhibitor, PI103 | PI-103 | 3-...)
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3K delta (unknown origin) using PIP2 as substrate after 1 hr by kinase-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM25045(CHEMBL538346 | mTOR Inhibitor, PI103 | PI-103 | 3-...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human recombinant PI3K delta by scintillation proximity radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50148942(CHEMBL3769902)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of PI3K alpha (unknown origin) using PIP2 as substrate after 1 hr by kinase-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM25045(CHEMBL538346 | mTOR Inhibitor, PI103 | PI-103 | 3-...)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of human recombinant PI3K alpha by scintillation proximity radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM25045(CHEMBL538346 | mTOR Inhibitor, PI103 | PI-103 | 3-...)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of PI3K alpha (unknown origin) using PIP2 as substrate after 1 hr by kinase-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50149057(CHEMBL3771212)
Affinity DataIC50: 11nMAssay Description:Inhibition of PI3K alpha (unknown origin) using PIP2 as substrate after 1 hr by kinase-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50148942(CHEMBL3769902)
Affinity DataIC50: 13nMAssay Description:Inhibition of PI3K beta (unknown origin) after 1 hr by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50149154(CHEMBL3771146)
Affinity DataIC50: 13nMAssay Description:Inhibition of PI3K alpha (unknown origin) using PIP2 as substrate after 1 hr by kinase-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM25045(CHEMBL538346 | mTOR Inhibitor, PI103 | PI-103 | 3-...)
Affinity DataIC50: 15nMAssay Description:Inhibition of human recombinant PI3K gamma by scintillation proximity radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM25045(CHEMBL538346 | mTOR Inhibitor, PI103 | PI-103 | 3-...)
Affinity DataIC50: 16nMAssay Description:Inhibition of mTOR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM25045(CHEMBL538346 | mTOR Inhibitor, PI103 | PI-103 | 3-...)
Affinity DataIC50: 21nMAssay Description:Inhibition of PI3K beta (unknown origin) after 1 hr by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM25045(CHEMBL538346 | mTOR Inhibitor, PI103 | PI-103 | 3-...)
Affinity DataIC50: 21nMAssay Description:Inhibition of PI3K beta (unknown origin) after 1 hr by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50149153(CHEMBL3769845)
Affinity DataIC50: 31nMAssay Description:Inhibition of PI3K alpha (unknown origin) using PIP2 as substrate after 1 hr by kinase-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50149055(CHEMBL3771347)
Affinity DataIC50: 33nMAssay Description:Inhibition of PI3K alpha (unknown origin) using PIP2 as substrate after 1 hr by kinase-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50149210(CHEMBL3769994)
Affinity DataIC50: 49nMAssay Description:Inhibition of PI3K alpha (unknown origin) using PIP2 as substrate after 1 hr by kinase-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50148942(CHEMBL3769902)
Affinity DataIC50: 50nMAssay Description:Inhibition of PI3K delta (unknown origin) using PIP2 as substrate after 1 hr by kinase-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM25045(CHEMBL538346 | mTOR Inhibitor, PI103 | PI-103 | 3-...)
Affinity DataIC50: 51nMAssay Description:Inhibition of PI3K gamma (unknown origin) after 1 hr by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50148942(CHEMBL3769902)
Affinity DataIC50: 64nMAssay Description:Inhibition of PI3K gamma (unknown origin) after 1 hr by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50149049(CHEMBL3771060)
Affinity DataIC50: 74nMAssay Description:Inhibition of PI3K alpha (unknown origin) using PIP2 as substrate after 1 hr by kinase-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50148942(CHEMBL3769902)
Affinity DataIC50: 78nMAssay Description:Inhibition of mTOR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50149056(CHEMBL3771348)
Affinity DataIC50: 142nMAssay Description:Inhibition of human recombinant PI3K alpha by scintillation proximity radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50149047(CHEMBL3770469)
Affinity DataIC50: 232nMAssay Description:Inhibition of human recombinant PI3K alpha by scintillation proximity radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50149046(CHEMBL3770892)
Affinity DataIC50: 393nMAssay Description:Inhibition of human recombinant PI3K alpha by scintillation proximity radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50149052(CHEMBL3770661)
Affinity DataIC50: 406nMAssay Description:Inhibition of human recombinant PI3K alpha by scintillation proximity radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50149156(CHEMBL3771094)
Affinity DataIC50: 419nMAssay Description:Inhibition of PI3K alpha (unknown origin) using PIP2 as substrate after 1 hr by kinase-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50149042(CHEMBL3769535)
Affinity DataIC50: 609nMAssay Description:Inhibition of human recombinant PI3K alpha by scintillation proximity radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50149102(CHEMBL3770944)
Affinity DataIC50: 778nMAssay Description:Inhibition of human recombinant PI3K alpha by scintillation proximity radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50149155(CHEMBL3770226)
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of human recombinant PI3K alpha by scintillation proximity radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50149048(CHEMBL3770633)
Affinity DataIC50: 2.17E+3nMAssay Description:Inhibition of PI3K alpha (unknown origin) using PIP2 as substrate after 1 hr by kinase-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50149045(CHEMBL3770985)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3K alpha (unknown origin) using PIP2 as substrate after 1 hr by kinase-Glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50149152(CHEMBL3770928)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant PI3K alpha by scintillation proximity radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
LigandPNGBDBM50149209(CHEMBL3771166)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant PI3K alpha by scintillation proximity radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed