Compile Data Set for Download or QSAR
Report error Found 237 Enz. Inhib. hit(s) with all data for entry = 50046959
Target5-hydroxytryptamine receptor 1A(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140055(CHEMBL3754166)
Affinity DataKi:  10nMAssay Description:Binding affinity to 5-HT 1A (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140053(CHEMBL3754496)
Affinity DataKi:  17nMAssay Description:Binding affinity to 5-HT 2B (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50435344(CHEMBL2391541)
Affinity DataKi:  19nMAssay Description:Binding affinity to 5-HT 1A (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50435344(CHEMBL2391541)
Affinity DataKi:  20nMAssay Description:Binding affinity to 5-HT 1A (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140054(CHEMBL3752900)
Affinity DataKi:  30nMAssay Description:Binding affinity to 5-HT 2B (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140056(CHEMBL3753318)
Affinity DataKi:  32nMAssay Description:Binding affinity to 5-HT 1A (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140053(CHEMBL3754496)
Affinity DataKi:  36nMAssay Description:Binding affinity to SERT (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140054(CHEMBL3752900)
Affinity DataKi:  41nMAssay Description:Binding affinity to SERT (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140055(CHEMBL3754166)
Affinity DataKi:  49nMAssay Description:Binding affinity to 5-HT 7 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140055(CHEMBL3754166)
Affinity DataKi:  52nMAssay Description:Binding affinity to 5-HT 2B (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50435344(CHEMBL2391541)
Affinity DataKi:  59nMAssay Description:Binding affinity to 5-HT 2B (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140054(CHEMBL3752900)
Affinity DataKi:  59nMAssay Description:Binding affinity to 5-HT 1A (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140056(CHEMBL3753318)
Affinity DataKi:  60nMAssay Description:Binding affinity to 5-HT 2B (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140058(CHEMBL3752576)
Affinity DataKi:  62nMAssay Description:Binding affinity to 5-HT 2B (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140054(CHEMBL3752900)
Affinity DataKi:  69nMAssay Description:Binding affinity to 5-HT 6 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140056(CHEMBL3753318)
Affinity DataKi:  74nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140054(CHEMBL3752900)
Affinity DataKi:  74nMAssay Description:Binding affinity to 5-HT 7 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140053(CHEMBL3754496)
Affinity DataKi:  74nMAssay Description:Binding affinity to 5-HT 6 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140053(CHEMBL3754496)
Affinity DataKi:  79nMAssay Description:Binding affinity to 5-HT 1A (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140053(CHEMBL3754496)
Affinity DataKi:  79nMAssay Description:Binding affinity to histamine H1 receptor (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140054(CHEMBL3752900)
Affinity DataKi:  81nMAssay Description:Binding affinity to alpha-2A adrenergic receptor (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140055(CHEMBL3754166)
Affinity DataKi:  83nMAssay Description:Binding affinity to alpha-2A adrenergic receptor (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140053(CHEMBL3754496)
Affinity DataKi:  85nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50435344(CHEMBL2391541)
Affinity DataKi:  89nMAssay Description:Binding affinity to 5-HT 7 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140054(CHEMBL3752900)
Affinity DataKi:  98nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140055(CHEMBL3754166)
Affinity DataKi:  100nMAssay Description:Binding affinity to histamine H1 receptor (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50435344(CHEMBL2391541)
Affinity DataKi:  100nMAssay Description:Binding affinity to 5-HT 1D (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140058(CHEMBL3752576)
Affinity DataKi:  100nMAssay Description:Binding affinity to 5-HT 1A (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140058(CHEMBL3752576)
Affinity DataKi:  100nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50435344(CHEMBL2391541)
Affinity DataKi:  100nMAssay Description:Binding affinity to 5-HT 1D (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140054(CHEMBL3752900)
Affinity DataKi:  100nMAssay Description:Binding affinity to histamine H1 receptor (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140055(CHEMBL3754166)
Affinity DataKi:  102nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140053(CHEMBL3754496)
Affinity DataKi:  102nMAssay Description:Binding affinity to 5-HT 2C (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140053(CHEMBL3754496)
Affinity DataKi:  117nMAssay Description:Binding affinity to alpha-2A adrenergic receptor (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140053(CHEMBL3754496)
Affinity DataKi:  120nMAssay Description:Binding affinity to D3 dopamine receptor (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140058(CHEMBL3752576)
Affinity DataKi:  123nMAssay Description:Binding affinity to alpha-2A adrenergic receptor (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140055(CHEMBL3754166)
Affinity DataKi:  126nMAssay Description:Binding affinity to 5-HT 1D (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140058(CHEMBL3752576)
Affinity DataKi:  126nMAssay Description:Binding affinity to histamine H1 receptor (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140055(CHEMBL3754166)
Affinity DataKi:  126nMAssay Description:Binding affinity to SERT (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140055(CHEMBL3754166)
Affinity DataKi:  132nMAssay Description:Binding affinity to 5-HT 6 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140054(CHEMBL3752900)
Affinity DataKi:  141nMAssay Description:Binding affinity to D3 dopamine receptor (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140058(CHEMBL3752576)
Affinity DataKi:  151nMAssay Description:Binding affinity to SERT (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140056(CHEMBL3753318)
Affinity DataKi:  155nMAssay Description:Binding affinity to 5-HT 7 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50435344(CHEMBL2391541)
Affinity DataKi:  155nMAssay Description:Binding affinity to 5-HT 6 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140054(CHEMBL3752900)
Affinity DataKi:  170nMAssay Description:Binding affinity to alpha-2B adrenergic receptor (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140056(CHEMBL3753318)
Affinity DataKi:  195nMAssay Description:Binding affinity to alpha-2A adrenergic receptor (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140054(CHEMBL3752900)
Affinity DataKi:  204nMAssay Description:Binding affinity to 5-HT 2C (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50140054(CHEMBL3752900)
Affinity DataKi:  214nMAssay Description:Binding affinity to 5-HT 1D (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50435344(CHEMBL2391541)
Affinity DataKi:  214nMAssay Description:Binding affinity to alpha-2A adrenergic receptor (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
The Alexander Shulgin Research Institute

Curated by ChEMBL
LigandPNGBDBM50435344(CHEMBL2391541)
Affinity DataKi:  218nMAssay Description:Binding affinity to 5-HT 2A (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2017
Entry Details Article
PubMed
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