Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50046971
TargetIntegrin alpha-V/beta-3(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50235980(CHEMBL429876 | EMD-121974 | cyclo(Arg-Gly-Asp-D-Ph...)
Affinity DataIC50: 0.400nMAssay Description:Binding affinity to integrin alphav/beta3 heterodimer in human M21 cells assessed as inhibition of integrin-mediated human M21 cell adhesion to vitro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2017
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50140178(CHEMBL3754350)
Affinity DataIC50: 2.40nMAssay Description:Binding affinity to integrin alphav/beta3 heterodimer in human M21 cells assessed as inhibition of integrin-mediated human M21 cell adhesion to vitro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2017
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50140179(CHEMBL3753748)
Affinity DataIC50: 15nMAssay Description:Binding affinity to integrin alpha5/beta1 heterodimer in human K562 cells assessed as inhibition of integrin-mediated human K562 cell adhesion to fib...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2017
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50140177(CHEMBL3752070)
Affinity DataIC50: 20nMAssay Description:Binding affinity to integrin alphav/beta3 heterodimer (unknown origin) assessed as inhibition of integrin-mediated cell adhesion to vitronectinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2017
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50140178(CHEMBL3754350)
Affinity DataIC50: 26nMAssay Description:Binding affinity to integrin alpha5/beta1 heterodimer in human K562 cells assessed as inhibition of integrin-mediated human K562 cell adhesion to fib...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2017
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50140179(CHEMBL3753748)
Affinity DataIC50: 34nMAssay Description:Binding affinity to integrin alphav/beta3 heterodimer in human M21 cells assessed as inhibition of integrin-mediated human M21 cell adhesion to vitro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2017
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50140177(CHEMBL3752070)
Affinity DataIC50: 1.50E+3nMAssay Description:Binding affinity to integrin alpha5/beta1 heterodimer (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2017
Entry Details Article
PubMed