Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50047026
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataEC50:  5nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in CHO cells assessed as increase in intracellular calcium mobilization after 90 secs by Cal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144609(CHEMBL3759222)
Affinity DataEC50:  20nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in CHO cells assessed as increase in intracellular calcium mobilization after 90 secs by Cal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144618(CHEMBL3758534)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144619(CHEMBL3759785)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144614(CHEMBL3758884)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144609(CHEMBL3759222)
Affinity DataKi:  8.80nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144615(CHEMBL3759255)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144612(CHEMBL3759254)
Affinity DataKi:  9.60nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144617(CHEMBL3759440)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144616(CHEMBL3758338)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144610(CHEMBL3759228)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144611(CHEMBL3758491)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144613(CHEMBL3758753)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  313nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144618(CHEMBL3758534)
Affinity DataKi:  1.04E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144609(CHEMBL3759222)
Affinity DataKi:  1.55E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144614(CHEMBL3758884)
Affinity DataKi:  1.73E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144617(CHEMBL3759440)
Affinity DataKi:  1.79E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144616(CHEMBL3758338)
Affinity DataKi:  1.81E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144619(CHEMBL3759785)
Affinity DataKi:  1.93E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144615(CHEMBL3759255)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144613(CHEMBL3758753)
Affinity DataKi:  4.41E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144612(CHEMBL3759254)
Affinity DataKi:  4.72E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144611(CHEMBL3758491)
Affinity DataKi:  6.21E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50144610(CHEMBL3759228)
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMed