Compile Data Set for Download or QSAR
Report error Found 160 Enz. Inhib. hit(s) with all data for entry = 7124
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175369(8-[4-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phen...)
Affinity DataKi:  63nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175395(1,3-Dimethyl-8-[{3-(2-(dimethylaminoethylamino)-2-...)
Affinity DataKi:  75nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175398(1,3-Dimethyl-8-[4-methoxy-3-{2-(piperidin-1-yl)-2-...)
Affinity DataKi:  76nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175399(1,3-Dimethyl-8-[{3-(2-(hexamethyleneimin-1-yl)-2-o...)
Affinity DataKi:  94nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175368(1,3-Dimethyl-8-[4-{2-(dimethylaminoethylamino)-2-o...)
Affinity DataKi:  100nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175370(1,3-Dimethyl-8-[4-{2-(pyrrolidin-1-yl)-2-oxoethoxy...)
Affinity DataKi:  122nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175396(8-[{3-(2-(Diethylaminoethylamino)-2-oxoethoxy)-4-m...)
Affinity DataKi:  126nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175376(1,3-Dimethyl-8-[4-{2-(homoveratrylamino)-2-oxoetho...)
Affinity DataKi:  128nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175377(1,3-Dimethyl-8-[3-{2-(dimethylaminoethylamino)-2-o...)
Affinity DataKi:  163nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175364(1,3-Dimethyl-8-[4-(2-methoxy-2-oxoethoxy)-phenyl]x...)
Affinity DataKi:  170nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175371(1,3-Dimethyl-8-[4-{2-(piperidin-1-yl)-2-oxoethoxy}...)
Affinity DataKi:  178nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175378(8-[3-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phen...)
Affinity DataKi:  179nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175374(1,3-Dimethyl-8-[4-{2-(1-methylpiperazin-4-yl)-2-ox...)
Affinity DataKi:  193nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175380(1,3-Dimethyl-8-[3-{2-(piperidin-1-yl)]-2-oxoethoxy...)
Affinity DataKi:  209nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Panjab University

LigandPNGBDBM175368(1,3-Dimethyl-8-[4-{2-(dimethylaminoethylamino)-2-o...)
Affinity DataKi:  220nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175381(1,3-Dimethyl-8-[3-{2-(hexamethyleneimin-1-yl)-2-ox...)
Affinity DataKi:  226nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175379(1,3-Dimethyl-8-[3-{2-(pyrrolidin-1-yl)-2-oxoethoxy...)
Affinity DataKi:  237nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175397(1,3-Dimethyl-8-[4-methoxy-3-{2-(pyrrolidin-1-yl)-2...)
Affinity DataKi:  259nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175372(1,3-Dimethyl-8-[4-{2-(hexamethyleneimin-1-yl)-2-ox...)
Affinity DataKi:  273nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175373(1,3-Dimethyl-8-[4-{2-(morpholin-1-yl)-2-oxoethoxy}...)
Affinity DataKi:  283nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Panjab University

LigandPNGBDBM175369(8-[4-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phen...)
Affinity DataKi:  298nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Panjab University

LigandPNGBDBM175364(1,3-Dimethyl-8-[4-(2-methoxy-2-oxoethoxy)-phenyl]x...)
Affinity DataKi:  319nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175365(1,3-Dimethyl-8-[3-(2-methoxy-2-oxoethoxy)-phenyl]x...)
Affinity DataKi:  375nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Panjab University

LigandPNGBDBM175371(1,3-Dimethyl-8-[4-{2-(piperidin-1-yl)-2-oxoethoxy}...)
Affinity DataKi:  401nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Panjab University

LigandPNGBDBM175371(1,3-Dimethyl-8-[4-{2-(piperidin-1-yl)-2-oxoethoxy}...)
Affinity DataKi:  419nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Panjab University

LigandPNGBDBM175372(1,3-Dimethyl-8-[4-{2-(hexamethyleneimin-1-yl)-2-ox...)
Affinity DataKi:  443nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175400(1,3-Dimethyl-8-[4-methoxy-3-{(2-(morpholin-1-yl)-2...)
Affinity DataKi:  466nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Panjab University

LigandPNGBDBM175374(1,3-Dimethyl-8-[4-{2-(1-methylpiperazin-4-yl)-2-ox...)
Affinity DataKi:  499nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175384(1,3-Dimethyl-8-[3-{2-(imidazol-1-yl)-2-oxoethoxy}-...)
Affinity DataKi:  509nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Panjab University

LigandPNGBDBM175376(1,3-Dimethyl-8-[4-{2-(homoveratrylamino)-2-oxoetho...)
Affinity DataKi:  516nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175383(1,3-Dimethyl-8-[3-{2-(1-methylpiperazin-4-yl)-2-ox...)
Affinity DataKi:  561nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Panjab University

LigandPNGBDBM175372(1,3-Dimethyl-8-[4-{2-(hexamethyleneimin-1-yl)-2-ox...)
Affinity DataKi:  609nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175382(1,3-Dimethyl-8-[3-{2-(morpholin-1-yl)-2-oxoethoxy}...)
Affinity DataKi:  679nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Panjab University

LigandPNGBDBM175377(1,3-Dimethyl-8-[3-{2-(dimethylaminoethylamino)-2-o...)
Affinity DataKi:  683nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175401(1,3-Dimethyl-8-[4-methoxy-3-{2-(1-methylpiperazin-...)
Affinity DataKi:  685nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175387(8-[{4-(2-(Diethylaminoethylamino)-2-oxoethoxy)-3-m...)
Affinity DataKi:  692nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175367(1,3-Dimethyl-8-[{3-(2-methoxy-2-oxoethoxy)-4-metho...)
Affinity DataKi:  717nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175403(1,3-Dimethyl-8-[{3-(2-(homoveratrylamino)-2-oxoeth...)
Affinity DataKi:  772nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Panjab University

LigandPNGBDBM175370(1,3-Dimethyl-8-[4-{2-(pyrrolidin-1-yl)-2-oxoethoxy...)
Affinity DataKi:  796nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A3 [I248L](Human)
Panjab University

LigandPNGBDBM175399(1,3-Dimethyl-8-[{3-(2-(hexamethyleneimin-1-yl)-2-o...)
Affinity DataKi:  797nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175386(1,3-Dimethyl-8-[{4-(2-(dimethylaminoethylamino)-2-...)
Affinity DataKi:  821nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175394(1,3-Dimethyl-8-[{4-(2-(homoveratrylamino)-2-oxoeth...)
Affinity DataKi:  843nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Panjab University

LigandPNGBDBM175395(1,3-Dimethyl-8-[{3-(2-(dimethylaminoethylamino)-2-...)
Affinity DataKi:  847nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Panjab University

LigandPNGBDBM175368(1,3-Dimethyl-8-[4-{2-(dimethylaminoethylamino)-2-o...)
Affinity DataKi:  903nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Panjab University

LigandPNGBDBM175374(1,3-Dimethyl-8-[4-{2-(1-methylpiperazin-4-yl)-2-ox...)
Affinity DataKi:  954nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Panjab University

LigandPNGBDBM175369(8-[4-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phen...)
Affinity DataKi:  968nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Panjab University

LigandPNGBDBM175364(1,3-Dimethyl-8-[4-(2-methoxy-2-oxoethoxy)-phenyl]x...)
Affinity DataKi:  980nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Panjab University

LigandPNGBDBM175402(1,3-Dimethyl-8-[{3-(2-(imidazol-1-yl)-2-oxoethoxy)...)
Affinity DataKi:  1.12E+3nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Panjab University

LigandPNGBDBM175378(8-[3-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phen...)
Affinity DataKi:  1.22E+3nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Panjab University

LigandPNGBDBM175373(1,3-Dimethyl-8-[4-{2-(morpholin-1-yl)-2-oxoethoxy}...)
Affinity DataKi:  1.25E+3nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details Article
PubMed
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