Compile Data Set for Download or QSAR
Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50047319
TargetCholinesterase(Human)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160078(CHEMBL3787613)
Affinity DataIC50: 13nMAssay Description:Inhibition of human butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160078(CHEMBL3787613)
Affinity DataIC50: 14nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160250(CHEMBL3785472)
Affinity DataIC50: 21nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160255(CHEMBL3785189)
Affinity DataIC50: 22nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160077(CHEMBL3785861)
Affinity DataIC50: 23nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50004000(CHEMBL94 | physostigmine | Antilirium | Eserine | ...)
Affinity DataIC50: 32nMAssay Description:Inhibition of human acetylcholinesterase using acetylcholine iodide as substrate preincubated for 30 mins followed by substrate addition measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160247(CHEMBL3786119)
Affinity DataIC50: 34nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160249(CHEMBL3785181)
Affinity DataIC50: 40nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160076(CHEMBL3787116)
Affinity DataIC50: 44nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50004000(CHEMBL94 | physostigmine | Antilirium | Eserine | ...)
Affinity DataIC50: 78nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160254(CHEMBL3786737)
Affinity DataIC50: 83nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160266(CHEMBL3787106)
Affinity DataIC50: 96nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160268(CHEMBL3786381)
Affinity DataIC50: 106nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160267(CHEMBL3785533)
Affinity DataIC50: 115nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160263(CHEMBL3786599)
Affinity DataIC50: 199nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160260(CHEMBL3786761)
Affinity DataIC50: 208nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160264(CHEMBL3787432)
Affinity DataIC50: 231nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160259(CHEMBL3785401)
Affinity DataIC50: 238nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160262(CHEMBL3787015)
Affinity DataIC50: 251nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160252(CHEMBL3786979)
Affinity DataIC50: 374nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160265(CHEMBL3785143)
Affinity DataIC50: 474nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160251(CHEMBL3785766)
Affinity DataIC50: 531nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160256(CHEMBL3785190)
Affinity DataIC50: 565nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160257(CHEMBL3787554)
Affinity DataIC50: 723nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160077(CHEMBL3785861)
Affinity DataIC50: 852nMAssay Description:Inhibition of human acetylcholinesterase using acetylcholine iodide as substrate preincubated for 30 mins followed by substrate addition measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160261(CHEMBL3785495)
Affinity DataIC50: 875nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160076(CHEMBL3787116)
Affinity DataIC50: 1.61E+3nMAssay Description:Inhibition of human acetylcholinesterase using acetylcholine iodide as substrate preincubated for 30 mins followed by substrate addition measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160245(CHEMBL3785462)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160086(CHEMBL3786447)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160181(CHEMBL3786505)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160258(CHEMBL3787268)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160082(CHEMBL3785481)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160081(CHEMBL3786666)
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160275(CHEMBL3785561)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160088(CHEMBL3785229)
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160081(CHEMBL3786666)
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of human acetylcholinesterase using acetylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160237(CHEMBL3785644)
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160270(CHEMBL3786576)
Affinity DataIC50: 1.48E+4nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160083(CHEMBL3786655)
Affinity DataIC50: 1.53E+4nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160271(CHEMBL3786390)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160091(CHEMBL3786323)
Affinity DataIC50: 1.74E+4nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160139(CHEMBL3786589)
Affinity DataIC50: 2.26E+4nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160079(CHEMBL3786544)
Affinity DataIC50: 2.28E+4nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160253(CHEMBL3786556)
Affinity DataIC50: 3.62E+4nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160089(CHEMBL3785187)
Affinity DataIC50: 3.95E+4nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160244(CHEMBL3785808)
Affinity DataIC50: 3.99E+4nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160080(CHEMBL3787307)
Affinity DataIC50: 5.58E+4nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160276(CHEMBL3786978)
Affinity DataIC50: 5.60E+4nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160087(CHEMBL3787666)
Affinity DataIC50: 5.89E+4nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160085(CHEMBL3786843)
Affinity DataIC50: 6.32E+4nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMed
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