Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50047519
TargetOxysterols receptor LXR-beta(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50172624(CHEMBL3809494)
Affinity DataEC50:  7nMAssay Description:Agonist activity at LXRbeta (unknown origin) expressed in human H4 cells co-expressing ABCA1 promoter measured after 48 hrs by cell-based transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50172624(CHEMBL3809494)
Affinity DataEC50:  8nMAssay Description:Agonist activity at GST-tagged LXRbeta-LBD (unknown origin) by LanthaScreen TR-FRET liver X receptor coactivator assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at LXRalpha (unknown origin) expressed in human HepG2 cells co-expressing ABCA1 promoter measured after 48 hrs by cell-based transac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-beta(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at LXRbeta (unknown origin) expressed in human H4 cells co-expressing ABCA1 promoter measured after 48 hrs by cell-based transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-beta(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50172521(CHEMBL3809850)
Affinity DataEC50:  30nMAssay Description:Agonist activity at GST-tagged LXRbeta-LBD (unknown origin) by LanthaScreen TR-FRET liver X receptor coactivator assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-alpha(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50172624(CHEMBL3809494)
Affinity DataEC50:  41nMAssay Description:Agonist activity at GST-tagged LXRalpha-LBD (unknown origin) by LanthaScreen TR-FRET liver X receptor coactivator assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50172624(CHEMBL3809494)
Affinity DataEC50:  45nMAssay Description:Agonist activity at LXRalpha (unknown origin) expressed in human HepG2 cells co-expressing ABCA1 promoter measured after 48 hrs by cell-based transac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50172646(CHEMBL3809583)
Affinity DataEC50:  280nMAssay Description:Agonist activity at LXRalpha (unknown origin) expressed in human HepG2 cells co-expressing ABCA1 promoter measured after 48 hrs by cell-based transac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50172521(CHEMBL3809850)
Affinity DataEC50:  420nMAssay Description:Partial agonist activity at GST-tagged LXRalpha-LBD (unknown origin) by LanthaScreen TR-FRET liver X receptor coactivator assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-alpha(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50172538(CHEMBL3808992)
Affinity DataEC50:  500nMAssay Description:Agonist activity at LXRalpha (unknown origin) expressed in human HepG2 cells co-expressing ABCA1 promoter measured after 48 hrs by cell-based transac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50172538(CHEMBL3808992)
Affinity DataEC50:  550nMAssay Description:Agonist activity at LXRbeta (unknown origin) expressed in human H4 cells co-expressing ABCA1 promoter measured after 48 hrs by cell-based transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50172646(CHEMBL3809583)
Affinity DataEC50:  770nMAssay Description:Agonist activity at LXRbeta (unknown origin) expressed in human H4 cells co-expressing ABCA1 promoter measured after 48 hrs by cell-based transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50172521(CHEMBL3809850)
Affinity DataEC50:  830nMAssay Description:Partial agonist activity at LXRalpha (unknown origin) expressed in human HepG2 cells co-expressing ABCA1 promoter measured after 48 hrs by cell-based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-beta(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50172505(CHEMBL3809555)
Affinity DataEC50:  840nMAssay Description:Agonist activity at GST-tagged LXRbeta-LBD (unknown origin) by LanthaScreen TR-FRET liver X receptor coactivator assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50172646(CHEMBL3809583)
Affinity DataEC50:  940nMAssay Description:Agonist activity at GST-tagged LXRbeta-LBD (unknown origin) by LanthaScreen TR-FRET liver X receptor coactivator assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50172646(CHEMBL3809583)
Affinity DataEC50:  1.48E+3nMAssay Description:Agonist activity at GST-tagged LXRalpha-LBD (unknown origin) by LanthaScreen TR-FRET liver X receptor coactivator assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50172505(CHEMBL3809555)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at LXRalpha (unknown origin) expressed in human HepG2 cells co-expressing ABCA1 promoter measured after 48 hrs by cell-based transac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMed