Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50047346
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
Lebanese University

Curated by ChEMBL
LigandPNGBDBM50161326(CHEMBL3787023)
Affinity DataIC50: 324nMAssay Description:Inhibition of human recombinant GST tagged IKK2 expressed in baculovirus using Ser/Thr05 peptide as substrate after 60 mins by Z-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2017
Entry Details Article
PubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
Lebanese University

Curated by ChEMBL
LigandPNGBDBM50161273(CHEMBL3787275)
Affinity DataIC50: 579nMAssay Description:Inhibition of human recombinant GST tagged IKK2 expressed in baculovirus using Ser/Thr05 peptide as substrate after 60 mins by Z-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2017
Entry Details Article
PubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
Lebanese University

Curated by ChEMBL
LigandPNGBDBM25919(N-(2-aminoethyl)-3,12-dimethyl-2,5,8-triazatricycl...)
Affinity DataIC50: 644nMAssay Description:Inhibition of human recombinant GST tagged IKK2 expressed in baculovirus using Ser/Thr05 peptide as substrate after 60 mins by Z-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2017
Entry Details Article
PubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
Lebanese University

Curated by ChEMBL
LigandPNGBDBM50161329(CHEMBL3786867)
Affinity DataIC50: 773nMAssay Description:Inhibition of human recombinant GST tagged IKK2 expressed in baculovirus using Ser/Thr05 peptide as substrate after 60 mins by Z-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2017
Entry Details Article
PubMed