Compile Data Set for Download or QSAR
Report error Found 82 Enz. Inhib. hit(s) with all data for entry = 50047269
TargetProstaglandin E2 receptor EP3 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156530(CHEMBL3793009)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP3 receptor expressed in CHO cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156528(CHEMBL3794185)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP4 receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156529(CHEMBL3794226)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP4 receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156530(CHEMBL3793009)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP4 receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156539(CHEMBL3793892)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP4 receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156472(CHEMBL3793167)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP3 receptor expressed in CHO cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156473(CHEMBL3793724)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP3 receptor expressed in CHO cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156474(CHEMBL3793515)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP3 receptor expressed in CHO cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156491(CHEMBL3792668)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP3 receptor expressed in CHO cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156528(CHEMBL3794185)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP3 receptor expressed in CHO cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156529(CHEMBL3794226)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP3 receptor expressed in CHO cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156491(CHEMBL3792668)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP4 receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156539(CHEMBL3793892)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP3 receptor expressed in CHO cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156472(CHEMBL3793167)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP1 receptor expressed in CHO cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156473(CHEMBL3793724)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP1 receptor expressed in CHO cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156474(CHEMBL3793515)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP1 receptor expressed in CHO cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156491(CHEMBL3792668)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP1 receptor expressed in CHO cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156528(CHEMBL3794185)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP1 receptor expressed in CHO cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156529(CHEMBL3794226)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP1 receptor expressed in CHO cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156530(CHEMBL3793009)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP1 receptor expressed in CHO cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156539(CHEMBL3793892)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP1 receptor expressed in CHO cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156473(CHEMBL3793724)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human IP receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156472(CHEMBL3793167)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human FP receptor expressed in Chem-1 cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156473(CHEMBL3793724)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human FP receptor expressed in Chem-1 cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156474(CHEMBL3793515)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human FP receptor expressed in Chem-1 cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156491(CHEMBL3792668)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human FP receptor expressed in Chem-1 cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156528(CHEMBL3794185)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human FP receptor expressed in Chem-1 cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156529(CHEMBL3794226)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human FP receptor expressed in Chem-1 cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156530(CHEMBL3793009)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human FP receptor expressed in Chem-1 cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156539(CHEMBL3793892)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human FP receptor expressed in Chem-1 cells assessed as intracellular Ca2+ level by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156472(CHEMBL3793167)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human IP receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156472(CHEMBL3793167)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP2 receptor expressed in HEK293 cells after 24 hrs beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156474(CHEMBL3793515)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human IP receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156491(CHEMBL3792668)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human IP receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156528(CHEMBL3794185)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human IP receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156529(CHEMBL3794226)
Affinity DataEC50:  5.30E+3nMAssay Description:Agonist activity at human IP receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156530(CHEMBL3793009)
Affinity DataEC50:  7.90E+3nMAssay Description:Agonist activity at human IP receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156539(CHEMBL3793892)
Affinity DataEC50:  4.90E+3nMAssay Description:Agonist activity at human IP receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156472(CHEMBL3793167)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP4 receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156473(CHEMBL3793724)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP4 receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156474(CHEMBL3793515)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human EP4 receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156534(CHEMBL3793809)
Affinity DataEC50:  3.90nMAssay Description:Agonist activity at human EP2 receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156544(CHEMBL3793209)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human EP2 receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156543(CHEMBL3793045)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at human EP2 receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156542(CHEMBL3793786)
Affinity DataEC50:  3.90nMAssay Description:Agonist activity at human EP2 receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156541(CHEMBL3794302)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at human EP2 receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156540(CHEMBL3793802)
Affinity DataEC50:  0.570nMAssay Description:Agonist activity at human EP2 receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156539(CHEMBL3793892)
Affinity DataEC50:  0.690nMAssay Description:Agonist activity at human EP2 receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156538(CHEMBL3794466)
Affinity DataEC50:  0.680nMAssay Description:Agonist activity at human EP2 receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50156537(CHEMBL3793020)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human EP2 receptor expressed in CHO cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
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