Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 50047695
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184446(CHEMBL3823961)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184416(CHEMBL3822825)
Affinity DataIC50: 51nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184418(CHEMBL3822572)
Affinity DataIC50: 54nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184419(CHEMBL3823445)
Affinity DataIC50: 54nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184442(CHEMBL3823351)
Affinity DataIC50: 62nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184444(CHEMBL3823394)
Affinity DataIC50: 65nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184414(CHEMBL3823131)
Affinity DataIC50: 70nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184415(CHEMBL3823222)
Affinity DataIC50: 122nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184412(CHEMBL3823274)
Affinity DataIC50: 147nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184441(CHEMBL3823817)
Affinity DataIC50: 160nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184412(CHEMBL3823274)
Affinity DataIC50: 222nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184413(CHEMBL3823956)
Affinity DataIC50: 230nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184410(CHEBI:71013 | E-2007 | E2007 | ER-155055-90 | Fyco...)
Affinity DataIC50: 243nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-3 assessed as inhibition of glutamate-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184413(CHEMBL3823956)
Affinity DataIC50: 353nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184414(CHEMBL3823131)
Affinity DataIC50: 360nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184410(CHEBI:71013 | E-2007 | E2007 | ER-155055-90 | Fyco...)
Affinity DataIC50: 485nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-2 assessed as inhibition of glutamate-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184417(CHEMBL3823247)
Affinity DataIC50: 615nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184410(CHEBI:71013 | E-2007 | E2007 | ER-155055-90 | Fyco...)
Affinity DataIC50: 623nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-4 assessed as inhibition of glutamate-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184410(CHEBI:71013 | E-2007 | E2007 | ER-155055-90 | Fyco...)
Affinity DataIC50: 1.18E+3nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184445(CHEMBL3824102)
Affinity DataIC50: 1.79E+3nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184443(CHEMBL3824269)
Affinity DataIC50: 2.82E+3nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184411(CHEMBL3823441)
Affinity DataIC50: 2.97E+3nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184417(CHEMBL3823247)
Affinity DataIC50: 4.67E+3nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184410(CHEBI:71013 | E-2007 | E2007 | ER-155055-90 | Fyco...)
Affinity DataIC50: 6.51E+3nMAssay Description:Antagonist activity at human iGluA1 receptor flip isoform expressed in CHO-S cells assessed as inhibition of glutamate-induced increase in intracellu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184415(CHEMBL3823222)
Affinity DataIC50: 8.68E+3nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184443(CHEMBL3824269)
Affinity DataIC50: 9.26E+3nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-2 assessed as inhibition of glutamate-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184416(CHEMBL3822825)
Affinity DataIC50: 9.26E+3nMAssay Description:Antagonist activity at human iGluA1 receptor flip isoform expressed in CHO-S cells assessed as inhibition of glutamate-induced increase in intracellu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184417(CHEMBL3823247)
Affinity DataIC50: 9.26E+3nMAssay Description:Antagonist activity at human iGluA1 receptor flip isoform expressed in CHO-S cells assessed as inhibition of glutamate-induced increase in intracellu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184441(CHEMBL3823817)
Affinity DataIC50: 9.26E+3nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-2 assessed as inhibition of glutamate-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184443(CHEMBL3824269)
Affinity DataIC50: 9.26E+3nMAssay Description:Antagonist activity at human iGluA1 receptor flip isoform expressed in CHO-S cells assessed as inhibition of glutamate-induced increase in intracellu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184441(CHEMBL3823817)
Affinity DataIC50: 9.26E+3nMAssay Description:Antagonist activity at human iGluA1 receptor flip isoform expressed in CHO-S cells assessed as inhibition of glutamate-induced increase in intracellu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184445(CHEMBL3824102)
Affinity DataIC50: 9.26E+3nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-2 assessed as inhibition of glutamate-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184445(CHEMBL3824102)
Affinity DataIC50: 9.26E+3nMAssay Description:Antagonist activity at human iGluA1 receptor flip isoform expressed in CHO-S cells assessed as inhibition of glutamate-induced increase in intracellu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184416(CHEMBL3822825)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184444(CHEMBL3823394)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184418(CHEMBL3822572)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184442(CHEMBL3823351)
Affinity DataIC50: 2.57E+4nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-2 assessed as inhibition of glutamate-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184444(CHEMBL3823394)
Affinity DataIC50: 6.85E+4nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-2 assessed as inhibition of glutamate-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184417(CHEMBL3823247)
Affinity DataIC50: 8.33E+4nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-2 assessed as inhibition of glutamate-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184418(CHEMBL3822572)
Affinity DataIC50: 8.33E+4nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-2 assessed as inhibition of glutamate-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184415(CHEMBL3823222)
Affinity DataIC50: 8.33E+4nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-2 assessed as inhibition of glutamate-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184416(CHEMBL3822825)
Affinity DataIC50: 8.33E+4nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-2 assessed as inhibition of glutamate-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184419(CHEMBL3823445)
Affinity DataIC50: 8.33E+4nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-2 assessed as inhibition of glutamate-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184411(CHEMBL3823441)
Affinity DataIC50: 8.33E+4nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-3 assessed as inhibition of glutamate-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184411(CHEMBL3823441)
Affinity DataIC50: 8.33E+4nMAssay Description:Antagonist activity at human iGluA1 receptor flip isoform expressed in CHO-S cells assessed as inhibition of glutamate-induced increase in intracellu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184411(CHEMBL3823441)
Affinity DataIC50: 8.33E+4nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-4 assessed as inhibition of glutamate-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184414(CHEMBL3823131)
Affinity DataIC50: 8.33E+4nMAssay Description:Antagonist activity at human iGluA1 receptor flip isoform expressed in CHO-S cells assessed as inhibition of glutamate-induced increase in intracellu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184415(CHEMBL3823222)
Affinity DataIC50: 8.33E+4nMAssay Description:Antagonist activity at human iGluA1 receptor flip isoform expressed in CHO-S cells assessed as inhibition of glutamate-induced increase in intracellu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184412(CHEMBL3823274)
Affinity DataIC50: 8.33E+4nMAssay Description:Antagonist activity at human iGluA1 receptor flip isoform expressed in CHO-S cells assessed as inhibition of glutamate-induced increase in intracellu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetGlutamate receptor 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50184413(CHEMBL3823956)
Affinity DataIC50: 8.33E+4nMAssay Description:Antagonist activity at human iGluA1 receptor flip isoform expressed in CHO-S cells assessed as inhibition of glutamate-induced increase in intracellu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
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