Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50047696
TargetVitamin D3 receptor(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50124417(1Alpha,25-Dihydroxy-22-Oxavitamin D3 | 22-Oxacalci...)
Affinity DataEC50:  0.855nMAssay Description:Activation of VDR in human Jurkat cells expressing lentiviral VDRE-luciferase vector assessed as VDRE-mediated transcriptional activity measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  3.90nMAssay Description:Activation of VDR in human Jurkat cells expressing lentiviral VDRE-luciferase vector assessed as VDRE-mediated transcriptional activity measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50184448(CHEMBL3822832)
Affinity DataEC50:  31nMAssay Description:Activation of VDR in human Jurkat cells expressing lentiviral VDRE-luciferase vector assessed as VDRE-mediated transcriptional activity measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50184448(CHEMBL3822832)
Affinity DataEC50:  117nMAssay Description:Activation of VDR in human HaCaT cells expressing lentiviral VDRE-luciferase vector assessed as VDRE-mediated transcriptional activity measured after...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50124417(1Alpha,25-Dihydroxy-22-Oxavitamin D3 | 22-Oxacalci...)
Affinity DataEC50:  145nMAssay Description:Activation of VDR in human Caco2 cells expressing lentiviral VDRE-luciferase vector assessed as VDRE-mediated transcriptional activity measured after...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50124417(1Alpha,25-Dihydroxy-22-Oxavitamin D3 | 22-Oxacalci...)
Affinity DataEC50:  160nMAssay Description:Activation of VDR in human HaCaT cells expressing lentiviral VDRE-luciferase vector assessed as VDRE-mediated transcriptional activity measured after...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50184448(CHEMBL3822832)
Affinity DataEC50:  172nMAssay Description:Activation of VDR in human Caco2 cells expressing lentiviral VDRE-luciferase vector assessed as VDRE-mediated transcriptional activity measured after...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50184447(CHEMBL3822994)
Affinity DataEC50:  175nMAssay Description:Activation of VDR in human HaCaT cells expressing lentiviral VDRE-luciferase vector assessed as VDRE-mediated transcriptional activity measured after...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50184447(CHEMBL3822994)
Affinity DataEC50:  203nMAssay Description:Activation of VDR in human Jurkat cells expressing lentiviral VDRE-luciferase vector assessed as VDRE-mediated transcriptional activity measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  223nMAssay Description:Activation of VDR in human Caco2 cells expressing lentiviral VDRE-luciferase vector assessed as VDRE-mediated transcriptional activity measured after...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50184447(CHEMBL3822994)
Affinity DataEC50:  241nMAssay Description:Activation of VDR in human Caco2 cells expressing lentiviral VDRE-luciferase vector assessed as VDRE-mediated transcriptional activity measured after...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  250nMAssay Description:Activation of VDR in human HaCaT cells expressing lentiviral VDRE-luciferase vector assessed as VDRE-mediated transcriptional activity measured after...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50184449(CHEMBL3823776)
Affinity DataEC50:  484nMAssay Description:Activation of VDR in human HaCaT cells expressing lentiviral VDRE-luciferase vector assessed as VDRE-mediated transcriptional activity measured after...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50184449(CHEMBL3823776)
Affinity DataEC50:  562nMAssay Description:Activation of VDR in human Caco2 cells expressing lentiviral VDRE-luciferase vector assessed as VDRE-mediated transcriptional activity measured after...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50184449(CHEMBL3823776)
Affinity DataEC50:  653nMAssay Description:Activation of VDR in human Jurkat cells expressing lentiviral VDRE-luciferase vector assessed as VDRE-mediated transcriptional activity measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2017
Entry Details Article
PubMed