Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50047338
TargetNuclear receptor ROR-alpha(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50108881(CHEMBL3596591)
Affinity DataEC50:  390nMAssay Description:Inverse agonist activity at human ROR-alpha transfected in HEK293T cells by Gal4 luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50108881(CHEMBL3596591)
Affinity DataEC50:  200nMAssay Description:Inverse agonist activity at human ROR-gamma transfected in HEK293T cells by Gal4 luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-beta(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50108881(CHEMBL3596591)
Affinity DataEC50:  1.10E+3nMAssay Description:Inverse agonist activity at human ROR-beta transfected in HEK293T cells by Gal4 luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161155(CHEMBL3793229)
Affinity DataIC50: 10nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161156(CHEMBL3793914)
Affinity DataIC50: 56nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161154(CHEMBL3793036)
Affinity DataIC50: 72nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161145(CHEMBL3793667)
Affinity DataIC50: 72nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161157(CHEMBL3792836)
Affinity DataIC50: 200nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataIC50: 204nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161110(CHEMBL3792639)
Affinity DataIC50: 210nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50108881(CHEMBL3596591)
Affinity DataIC50: 220nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161107(CHEMBL3793430)
Affinity DataIC50: 520nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161109(CHEMBL3793855)
Affinity DataIC50: 520nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161106(CHEMBL3792498)
Affinity DataIC50: 630nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50108880(CHEMBL3596640)
Affinity DataIC50: 710nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161104(CHEMBL3792627)
Affinity DataIC50: 910nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161158(CHEMBL1475054)
Affinity DataIC50: 1.47E+3nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161116(CHEMBL3794408)
Affinity DataIC50: 1.50E+3nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161102(CHEMBL3793170)
Affinity DataIC50: 1.90E+3nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161108(CHEMBL3793608)
Affinity DataIC50: 2.80E+3nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161114(CHEMBL3794390)
Affinity DataIC50: 3.20E+3nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161115(CHEMBL3793397)
Affinity DataIC50: 3.80E+3nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161144(CHEMBL3794039)
Affinity DataIC50: 4.20E+3nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161112(CHEMBL3793917)
Affinity DataIC50: 4.70E+3nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161098(CHEMBL3793232)
Affinity DataIC50: 6.40E+3nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161105(CHEMBL3792422)
Affinity DataIC50: 6.50E+3nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161111(CHEMBL3793822)
Affinity DataIC50: 7.80E+3nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161101(CHEMBL3793403)
Affinity DataIC50: 8.10E+3nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161113(CHEMBL3793995)
Affinity DataIC50: 1.00E+4nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161100(CHEMBL3793784)
Affinity DataIC50: 1.00E+4nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161099(CHEMBL3793422)
Affinity DataIC50: 1.00E+4nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50161103(CHEMBL3792473)
Affinity DataIC50: 1.00E+4nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Biogen

Curated by ChEMBL
LigandPNGBDBM50108914(CHEMBL3596596)
Affinity DataIC50: 1.30E+4nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2017
Entry Details Article
PubMed