Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50047707
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50185005(CHEMBL3823483)
Affinity DataIC50: 28nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using myelin basic protein as substrate incubated for 30 mins in presen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2017
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50185005(CHEMBL3823483)
Affinity DataIC50: 41nMAssay Description:Inhibition of GST-tagged human recombinant CLK1 expressed in Escherichia coli using RS peptide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDual specificity protein kinase CLK1(Human)
University of Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50185004(CHEMBL3823532)
Affinity DataIC50: 69nMAssay Description:Inhibition of GST-tagged human recombinant CLK1 expressed in Escherichia coli using RS peptide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2017
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50185006(CHEMBL3823505)
Affinity DataIC50: 180nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using myelin basic protein as substrate incubated for 30 mins in presen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2017
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50185006(CHEMBL3823505)
Affinity DataIC50: 190nMAssay Description:Inhibition of GST-tagged human recombinant CLK1 expressed in Escherichia coli using RS peptide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50185004(CHEMBL3823532)
Affinity DataIC50: 620nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using myelin basic protein as substrate incubated for 30 mins in presen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50185005(CHEMBL3823483)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of GST-tagged human recombinant CDK5/p25 expressed in Escherichia coli using histone H1 as substrate incubated for 30 mins in presence of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50185004(CHEMBL3823532)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant CDK5/p25 expressed in Escherichia coli using histone H1 as substrate incubated for 30 mins in presence of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50185006(CHEMBL3823505)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant CDK5/p25 expressed in Escherichia coli using histone H1 as substrate incubated for 30 mins in presence of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2017
Entry Details Article
PubMed