Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50010186
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50529668(Enobosarm | Gtx-024 | MK-2866 | Ostarine | US10806...)
Affinity DataIC50: 36nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535824(CHEMBL4575144)
Affinity DataIC50: 49nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535836(CHEMBL4558169)
Affinity DataIC50: 59nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535830(CHEMBL4523011)
Affinity DataIC50: 72nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535839(CHEMBL4577418)
Affinity DataIC50: 80nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535835(CHEMBL4547536)
Affinity DataIC50: 111nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535841(CHEMBL4529395)
Affinity DataIC50: 123nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535837(CHEMBL4482919)
Affinity DataIC50: 183nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535829(CHEMBL4529026)
Affinity DataIC50: 198nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535825(CHEMBL4572299)
Affinity DataIC50: 245nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535834(CHEMBL4532289)
Affinity DataIC50: 265nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535826(CHEMBL4581453)
Affinity DataIC50: 280nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535827(CHEMBL4580745)
Affinity DataIC50: 332nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50425732(Xtandi | ENZALUTAMIDE | US10053433, FC 4.129 | US1...)
Affinity DataIC50: 361nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535840(CHEMBL4533483)
Affinity DataIC50: 402nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535843(CHEMBL4589154)
Affinity DataIC50: 407nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535823(CHEMBL4483683)
Affinity DataIC50: 425nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM18678(CHEMBL63560 | (2R)-N-[4-cyano-3-(trifluoromethyl)p...)
Affinity DataIC50: 490nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535828(CHEMBL4519421)
Affinity DataIC50: 625nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535842(CHEMBL4572778)
Affinity DataIC50: 625nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535831(CHEMBL4516292)
Affinity DataIC50: 736nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535832(CHEMBL4585541)
Affinity DataIC50: 775nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535833(CHEMBL4521612)
Affinity DataIC50: 777nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535844(CHEMBL4537113)
Affinity DataIC50: 811nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535845(CHEMBL4549022)
Affinity DataIC50: 1.07E+3nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
School of Pharmacy and Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50535838(CHEMBL4556247)
Affinity DataIC50: 2.17E+3nMAssay Description:Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed