Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50047433
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50118225(ARL 69931MX | Adenosine triphosphate derivative | ...)
Affinity DataIC50: 0.398nMAssay Description:Antagonist activity at P2Y12 receptor in human platelets assessed as inhibition of ADP-induced platelet aggregation by turbidimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50167270(CHEMBL1160364)
Affinity DataIC50: 0.794nMAssay Description:Antagonist activity at P2Y12 receptor in human platelets assessed as inhibition of ADP-induced platelet aggregation by turbidimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50167271(CHEMBL3798413)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at P2Y12 receptor in human platelets assessed as inhibition of ADP-induced platelet aggregation by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50167271(CHEMBL3798413)
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]-2-Mes-ADP from human P2Y12 receptor by beta-counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50118223(CHEMBL336292 | CHEMBL369928 | AR-C67085 | Adenosin...)
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at P2Y12 receptor in human platelets assessed as inhibition of ADP-induced platelet aggregation by turbidimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50397205(AR-C126532XX | AZD-6140 | AZD6140 | BRILINTA | TIC...)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50167273(CHEMBL3797316)
Affinity DataIC50: 5.30nMAssay Description:Displacement of [3H]-2-Mes-ADP from human P2Y12 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50167273(CHEMBL3797316)
Affinity DataIC50: 8.30nMAssay Description:Antagonist activity at P2Y12 receptor in human washed platelets assessed as inhibition of ADP-induced platelet aggregation measured for 5 mins by lig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50397204(ELINOGREL)
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]-2-Mes-ADP from human P2Y12 receptor in platelets by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50167272(CHEMBL3798029)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50397203(CHEMBL2172275)
Affinity DataIC50: 29nMAssay Description:Displacement of [3H]-2-Mes-ADP from human P2Y12 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50436962(CHEMBL2402264)
Affinity DataIC50: 40nMAssay Description:Binding affinity to P2Y12 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50439270(CHEMBL2419497)
Affinity DataIC50: 60nMAssay Description:Binding affinity to P2Y12 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50436962(CHEMBL2402264)
Affinity DataIC50: 70nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50439270(CHEMBL2419497)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50397203(CHEMBL2172275)
Affinity DataIC50: 130nMAssay Description:Antagonist activity at P2Y12 receptor in human washed platelets assessed as inhibition of ADP-induced platelet aggregation measured for 5 mins by lig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50167272(CHEMBL3798029)
Affinity DataIC50: 440nMAssay Description:Binding affinity to P2Y12 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50397204(ELINOGREL)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at P2Y12 receptor in human platelets assessed as inhibition of ADP-induced platelet aggregation by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50366480(ATP | ADENOSINE TRIPHOSPHATE)
Affinity DataIC50: 2.51E+5nMAssay Description:Antagonist activity at P2Y12 receptor in human platelets assessed as inhibition of ADP-induced platelet aggregation by turbidimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Galecto Biotech

Curated by ChEMBL
LigandPNGBDBM50167269(CHEMBL1160356)
Affinity DataIC50: 3.16E+5nMAssay Description:Antagonist activity at P2Y12 receptor in human platelets assessed as inhibition of ADP-induced platelet aggregation by turbidimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed