Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50047434
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167278(CHEMBL3800236)
Affinity DataEC50:  32nMAssay Description:Inhibition of human MetAP2 in HUVEC cells assessed as accumulation of N-Met 14-3-3gamma after 24 hrs by western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167279(CHEMBL3799090)
Affinity DataEC50:  20nMAssay Description:Inhibition of human MetAP2 in HUVEC cells assessed as accumulation of N-Met 14-3-3gamma after 24 hrs by western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167280(CHEMBL3797259)
Affinity DataEC50:  2.00E+3nMAssay Description:Inhibition of human MetAP2 in HUVEC cells assessed as accumulation of N-Met 14-3-3gamma after 24 hrs by western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167281(CHEMBL3799796)
Affinity DataEC50:  25nMAssay Description:Inhibition of human MetAP2 in HUVEC cells assessed as accumulation of N-Met 14-3-3gamma after 24 hrs by western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167285(CHEMBL3797780)
Affinity DataEC50:  251nMAssay Description:Inhibition of human MetAP2 in HUVEC cells assessed as accumulation of N-Met 14-3-3gamma after 24 hrs by western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167274(CHEMBL3797399)
Affinity DataEC50:  13nMAssay Description:Inhibition of human MetAP2 in HUVEC cells assessed as accumulation of N-Met 14-3-3gamma after 24 hrs by western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167275(CHEMBL3798249)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of human MetAP2 in HUVEC cells assessed as accumulation of N-Met 14-3-3gamma after 24 hrs by western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167276(CHEMBL3798844)
Affinity DataEC50:  1.26E+3nMAssay Description:Inhibition of human MetAP2 in HUVEC cells assessed as accumulation of N-Met 14-3-3gamma after 24 hrs by western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167277(CHEMBL3797386)
Affinity DataEC50:  100nMAssay Description:Inhibition of human MetAP2 in HUVEC cells assessed as accumulation of N-Met 14-3-3gamma after 24 hrs by western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167275(CHEMBL3798249)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167274(CHEMBL3797399)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167280(CHEMBL3797259)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167279(CHEMBL3799090)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167276(CHEMBL3798844)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167278(CHEMBL3800236)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167281(CHEMBL3799796)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167285(CHEMBL3797780)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167277(CHEMBL3797386)
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167276(CHEMBL3798844)
Affinity DataIC50: 50nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167320(CHEMBL3797508)
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167275(CHEMBL3798249)
Affinity DataIC50: 63nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167318(CHEMBL3797789)
Affinity DataIC50: 79nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167277(CHEMBL3797386)
Affinity DataIC50: 126nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167278(CHEMBL3800236)
Affinity DataIC50: 158nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167319(CHEMBL3797549)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167274(CHEMBL3797399)
Affinity DataIC50: 3.16E+3nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167280(CHEMBL3797259)
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167279(CHEMBL3799090)
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167281(CHEMBL3799796)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167285(CHEMBL3797780)
Affinity DataIC50: 5.01E+4nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed