Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50047764
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188633(CHEMBL3827045)
Affinity DataIC50: 99nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic VEGFR2 (789 to 1356 residues) expressed in baculovirus expression system incubated for 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188634(CHEMBL3828416)
Affinity DataIC50: 120nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic VEGFR2 (789 to 1356 residues) expressed in baculovirus expression system incubated for 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataIC50: 140nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic VEGFR2 (789 to 1356 residues) expressed in baculovirus expression system incubated for 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188632(CHEMBL3827784)
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic VEGFR2 (789 to 1356 residues) expressed in baculovirus expression system incubated for 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188635(CHEMBL3827098)
Affinity DataIC50: 330nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic VEGFR2 (789 to 1356 residues) expressed in baculovirus expression system incubated for 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM20607((2-{4-[(1Z)-1,2-diphenylbut-1-en-1-yl]phenoxy}ethy...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188628(CHEMBL3827137)
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic VEGFR2 (789 to 1356 residues) expressed in baculovirus expression system incubated for 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188632(CHEMBL3827784)
Affinity DataIC50: 3.40E+3nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188629(CHEMBL3827870)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic VEGFR2 (789 to 1356 residues) expressed in baculovirus expression system incubated for 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188634(CHEMBL3828416)
Affinity DataIC50: 6.70E+3nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188633(CHEMBL3827045)
Affinity DataIC50: 7.20E+3nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188635(CHEMBL3827098)
Affinity DataIC50: 7.60E+3nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188630(CHEMBL3828208)
Affinity DataIC50: 1.06E+4nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188627(CHEMBL3827692)
Affinity DataIC50: 1.77E+4nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188628(CHEMBL3827137)
Affinity DataIC50: 1.87E+4nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188631(CHEMBL3827200)
Affinity DataIC50: 1.98E+4nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188624(CHEMBL3827152)
Affinity DataIC50: 2.33E+4nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188629(CHEMBL3827870)
Affinity DataIC50: 2.44E+4nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188626(CHEMBL3827034)
Affinity DataIC50: 2.49E+4nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188601(CHEMBL3827633)
Affinity DataIC50: 3.52E+4nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188603(CHEMBL3828117)
Affinity DataIC50: 3.83E+4nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188606(CHEMBL3828422)
Affinity DataIC50: 3.94E+4nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188605(CHEMBL3827193)
Affinity DataIC50: 3.98E+4nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188604(CHEMBL3827286)
Affinity DataIC50: 4.03E+4nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188602(CHEMBL3827876)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50188625(CHEMBL3827018)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2017
Entry Details Article
PubMed