Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50047500
TargetEstrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50171495(CHEMBL3805318)
Affinity DataIC50: 0.0900nMAssay Description:Antagonist activity at ERalpha (unknown origin) transfected in 17beta-estradiol induced-HEK293 cells assessed as inhibition of estradiol-mediated pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM19441(Evista | CHEMBL81 | Keoxifene | Raloxifene, 6 | RA...)
Affinity DataIC50: 0.470nMAssay Description:Displacement of Fluormone ES2 from human recombinant full length untagged-ERalpha by fluorescence polarization competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50171494(CHEMBL3806167)
Affinity DataIC50: 0.680nMAssay Description:Antagonist activity at ERalpha (unknown origin) transfected in 17beta-estradiol induced-HEK293 cells assessed as inhibition of estradiol-mediated pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50171499(CHEMBL3805385)
Affinity DataIC50: 1.80nMAssay Description:Displacement of Fluormone ES2 from human recombinant full length untagged-ERalpha by fluorescence polarization competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50171495(CHEMBL3805318)
Affinity DataIC50: 5.90nMAssay Description:Displacement of Fluormone ES2 from human recombinant full length untagged-ERalpha by fluorescence polarization competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50171498(CHEMBL3805025)
Affinity DataIC50: 11nMAssay Description:Displacement of Fluormone ES2 from human recombinant full length untagged-ERalpha by fluorescence polarization competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50171497(CHEMBL3804907)
Affinity DataIC50: 28nMAssay Description:Displacement of Fluormone ES2 from human recombinant full length untagged-ERalpha by fluorescence polarization competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50171494(CHEMBL3806167)
Affinity DataIC50: 40nMAssay Description:Displacement of Fluormone ES2 from human recombinant full length untagged-ERalpha by fluorescence polarization competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50171493(CHEMBL3805170)
Affinity DataIC50: 49nMAssay Description:Displacement of Fluormone ES2 from human recombinant full length untagged-ERalpha by fluorescence polarization competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50171492(CHEMBL3805921)
Affinity DataIC50: 61nMAssay Description:Displacement of Fluormone ES2 from human recombinant full length untagged-ERalpha by fluorescence polarization competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2017
Entry Details Article
PubMed