Compile Data Set for Download or QSAR
Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 50047614
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178979(CHEMBL3813796)
Affinity DataIC50: 99nMAssay Description:Antagonist activity at human 5-HT2B receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178978(CHEMBL3815112)
Affinity DataIC50: 135nMAssay Description:Antagonist activity at human 5-HT2B receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178980(CHEMBL3813726)
Affinity DataIC50: 326nMAssay Description:Antagonist activity at human 5-HT2B receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178978(CHEMBL3815112)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50001775(cid_5074 | Ritanserine | 6-(2-{4-[Bis-(4-fluoro-ph...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]mesulergine from human 5-HT2C receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178979(CHEMBL3813796)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178980(CHEMBL3813726)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178981(CHEMBL3813855)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178973(CHEMBL3815066)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178964(CHEMBL3814737)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2A receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178969(CHEMBL3814821)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178977(CHEMBL3814559)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178968(CHEMBL3815000)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM82272(SB 200646 | SB200646a)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178963(CHEMBL3735756)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178979(CHEMBL3813796)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2A receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178966(CHEMBL3814485)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178967(CHEMBL3813789)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178965(CHEMBL3814708)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178980(CHEMBL3813726)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2A receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178978(CHEMBL3815112)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2A receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178981(CHEMBL3813855)
Affinity DataKi:  68nMAssay Description:Displacement of [3H]mesulergine from human 5-HT2C receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178981(CHEMBL3813855)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2A receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178978(CHEMBL3815112)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]mesulergine from human 5-HT2C receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178979(CHEMBL3813796)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]mesulergine from human 5-HT2C receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178973(CHEMBL3815066)
Affinity DataKi:  103nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2A receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178980(CHEMBL3813726)
Affinity DataKi:  124nMAssay Description:Displacement of [3H]mesulergine from human 5-HT2C receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178969(CHEMBL3814821)
Affinity DataKi:  125nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2A receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178964(CHEMBL3814737)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]mesulergine from human 5-HT2C receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178973(CHEMBL3815066)
Affinity DataKi:  143nMAssay Description:Displacement of [3H]mesulergine from human 5-HT2C receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178977(CHEMBL3814559)
Affinity DataKi:  154nMAssay Description:Displacement of [3H]mesulergine from human 5-HT2C receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178963(CHEMBL3735756)
Affinity DataKi:  165nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2A receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178968(CHEMBL3815000)
Affinity DataKi:  167nMAssay Description:Displacement of [3H]mesulergine from human 5-HT2C receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178977(CHEMBL3814559)
Affinity DataKi:  169nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2A receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178968(CHEMBL3815000)
Affinity DataKi:  185nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2A receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178964(CHEMBL3814737)
Affinity DataKi:  185nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2A receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178969(CHEMBL3814821)
Affinity DataKi:  206nMAssay Description:Displacement of [3H]mesulergine from human 5-HT2C receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178966(CHEMBL3814485)
Affinity DataKi:  219nMAssay Description:Displacement of [3H]mesulergine from human 5-HT2C receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178966(CHEMBL3814485)
Affinity DataKi:  221nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2A receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178967(CHEMBL3813789)
Affinity DataKi:  224nMAssay Description:Displacement of [3H]mesulergine from human 5-HT2C receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178965(CHEMBL3814708)
Affinity DataKi:  235nMAssay Description:Displacement of [3H]mesulergine from human 5-HT2C receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178967(CHEMBL3813789)
Affinity DataKi:  288nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2A receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178965(CHEMBL3814708)
Affinity DataKi:  365nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2A receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50178963(CHEMBL3735756)
Affinity DataKi:  399nMAssay Description:Displacement of [3H]mesulergine from human 5-HT2C receptor measured after 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed